SCHEMBL5565766

SCHEMBL5565766

O=S(=O)(Cl)c1cc(C(F)(F)F)cc(C(F)(F)F)c1.O=S(=O)(Cl)c1ccc(-c2ccccc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 2/20 0.48
ALDH1A1 P00352 2/20 0.47
HSD17B10 Q99714 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
ACLY P53396 4/20 0.45
MAPT P10636 2/20 0.44
PTPN1 P18031 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
RXRA P19793 1/20 0.42
RXRB P28702 1/20 0.42
RXRG P48443 1/20 0.42
MMP2 P08253 2/20 0.42
MMP9 P14780 2/20 0.42
MMP8 P22894 2/20 0.42
MMP12 P39900 1/20 0.42
MMP14 P50281 1/20 0.42
PDPK1 O15530 1/20 0.42
CA1 P00915 2/20 0.42
CA2 P00918 2/20 0.42
CA12 O43570 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14120499 0.86 RXRA (0.51) KIF11ALDH1A1HSD17B10TDP1RXRA
SCHEMBL5553604 0.85 PTGES2 (0.44) KIF11ALDH1A1HSD17B10TDP1ACLY
SCHEMBL7538033 0.84 KIF11 (0.47) KIF11ALDH1A1HSD17B10TDP1MAPT
SCHEMBL67742 0.82 CES2 (0.48) KIF11ALDH1A1HSD17B10TDP1MAPT
SCHEMBL3071920 0.81 KIF11 (0.66) KIF11MMP2MMP9PDPK1MMP1
SCHEMBL21993320 0.80 ALDH1A1 (0.71) ALDH1A1HSD17B10TDP1MMP2MMP14
SCHEMBL48861 0.80 ALDH1A1 (0.71) ALDH1A1HSD17B10TDP1MMP2MMP14
Hydrochloric Acid SCHEMBL5174554 0.78 ALDH1A1 (0.68) ALDH1A1HSD17B10TDP1MMP2MMP12
SCHEMBL14120723 0.75 CA1 (0.45) KIF11ALDH1A1HSD17B10TDP1ACLY
SCHEMBL9996829 0.75 KIF11 (0.54) KIF11ACLYPTPN1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1610753-A4 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC (US) 2007-07-04 EP disclosed
EP-1610753-A2 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC. (US) 2006-01-04 EP disclosed
WO-2004073634-A2 PHENYLENEDIAMINE UROTENSIN-II RECEPTOR ANTAGONISTS AND CCR-9 ANTAGONISTS ENCYSIVE PHARMACEUTICALS INC. (US) 2004-09-02 WO disclosed