SCHEMBL5583472

SCHEMBL5583472

Fc1ccc(-c2cc(F)c3c(c2)C[CH]O3)cc1

nearest known ligand 0.34

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.34
TDP2 O95551 1/20 0.34
CYP11B2 P19099 4/20 0.33
KDM1A O60341 2/20 0.33
CYP17A1 P05093 2/20 0.31
CYP11B1 P15538 3/20 0.31
MAOB P27338 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27723761 0.76 PTGS2 (0.35) CYP3A4CYP11B2
SCHEMBL4596976 0.69 PARP1 (0.44) KDM1A
SCHEMBL4596968 0.69 KDM1A (0.36) CYP3A4CYP11B2KDM1ACYP17A1CYP11B1
SCHEMBL4234781 0.66 PRKAB2 (0.53) KDM1AMAOB
SCHEMBL27723664 0.66 AQP1 (0.36) TDP2
SCHEMBL4230938 0.65 PRKAB2 (0.43) KDM1AMAOB
SCHEMBL2944704 0.65 BCL2L1 (0.48) CYP11B2CYP11B1MAOB
SCHEMBL19423241 0.65 BCL2L1 (0.48) CYP11B2CYP11B1MAOB
SCHEMBL4964977 0.64 TDP2 (0.33) TDP2
SCHEMBL4713338 0.62 GPBAR1 (0.34) TDP2CYP11B2CYP11B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2007509174-A 2007-04-12 JP claimed
EP-1675840-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS Wyeth a Corporation of the State of Delaware (US) 2006-07-05 EP claimed
WO-2005044812-A1 DIHYDROBENZOFURANYL ALKANAMINE DERIVATIVES AS 5HT2C AGONISTS WYETH A CORPORATION OF THE STATE OF DELAWARE (US) 2005-05-19 WO claimed