SCHEMBL5592387

SCHEMBL5592387

CN1CCN(c2cccc(F)c2CC2NCCN(c3ccc(C4CCOCC4)cc3)C2=O)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.35
ROCK2 O75116 1/20 0.35
FAAH O00519 2/20 0.34
BTK Q06187 5/20 0.33
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
MAPT P10636 1/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
HSD17B10 Q99714 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
PARP14 Q460N5 1/20 0.32
RAB9A P51151 1/20 0.32
DHFR P00374 1/20 0.32
RORC P51449 1/20 0.31
GRM2 Q14416 1/20 0.31
HTR1B P28222 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592318 0.86 MEN1 (0.36) BTKMEN1KMT2APOLBPARP14
SCHEMBL5592378 0.83 HSD11B1 (0.37) TRPV4ROCK2ALDH1A1POLBRORC
SCHEMBL5592321 0.80 SIGMAR1 (0.34) ROCK2ALDH1A1RORC
SCHEMBL5599159 0.78 ELANE (0.35) MAPTPARP14
SCHEMBL5592317 0.77 ALDH1A1 (0.37) TRPV4ROCK2ALDH1A1GAAALOX15
SCHEMBL5592394 0.72 MEN1 (0.35) BTKMEN1KMT2APOLBDHFR
SCHEMBL5809686 0.70 EGLN1 (0.39) ROCK2BTKALDH1A1GAAALOX15
SCHEMBL5592174 0.70 SLC6A2 (0.35) ALDH1A1MAPTHSD17B10MEN1KMT2A
SCHEMBL5739775 0.69 HSD11B1 (0.37) TRPV4ROCK2ALDH1A1HSD17B10POLB
SCHEMBL5812938 0.69 EGLN1 (0.36) BTKMEN1KMT2APOLBPARP14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007057742-A2 NOVEL PIPERAZINONE DERIVATIVES PFIZER PRODUCTS INC. (US) 2007-05-24 WO disclosed