SCHEMBL5592732

SCHEMBL5592732

CC(C)CNN(C(=O)c1cccc(CN2CCN(CCO)CC2)c1)c1nc(C#N)ncc1Cl

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.45
CTSS P25774 2/20 0.45
CTSK P43235 2/20 0.45
CTSB P07858 1/20 0.45
SRC P12931 2/20 0.35
HDAC3 O15379 2/20 0.35
HDAC4 P56524 2/20 0.35
HDAC1 Q13547 2/20 0.35
HDAC7 Q8WUI4 2/20 0.35
HDAC2 Q92769 2/20 0.35
HDAC10 Q969S8 2/20 0.35
HDAC11 Q96DB2 2/20 0.35
HDAC8 Q9BY41 2/20 0.35
HDAC6 Q9UBN7 2/20 0.35
HDAC9 Q9UKV0 2/20 0.35
HDAC5 Q9UQL6 2/20 0.35
WNT1 P04628 2/20 0.35
GSK3B P49841 2/20 0.35
DYRK1A Q13627 2/20 0.35
TNIK Q9UKE5 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592632 0.94 CTSL (0.45) CTSLCTSSCTSKCTSBHDAC3
SCHEMBL5593180 0.94 CTSL (0.45) CTSLCTSSCTSKCTSBHDAC3
SCHEMBL5592898 0.92 CTSL (0.43) CTSLCTSSCTSKCTSBHDAC3
SCHEMBL5592852 0.92 CTSL (0.43) CTSLCTSSCTSKCTSBWNT1
SCHEMBL5592899 0.84 CHEK1 (0.38) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5592870 0.83 CTSL (0.61) CTSLCTSSCTSKCTSBSRC
SCHEMBL5592735 0.82 CTSS (0.49) CTSLCTSSCTSKCTSB
SCHEMBL5592691 0.82 CTSS (0.49) CTSLCTSSCTSKCTSBHDAC1
Trifluoroacetic Acid SCHEMBL5592759 0.81 CTSL (0.47) CTSLCTSSCTSKCTSBCSF1R
Trifluoroacetic Acid SCHEMBL5592645 0.81 CTSS (0.47) CTSLCTSSCTSKCTSBCSF1R

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed