SCHEMBL5592852

SCHEMBL5592852

CC(C)CNN(C(=O)c1cccc(CN2CCCCC2)c1)c1nc(C#N)ncc1Cl

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43
CTSS P25774 1/20 0.43
CTSK P43235 1/20 0.43
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
HIF1A Q16665 1/20 0.40
PTGER1 P34995 2/20 0.38
WNT1 P04628 3/20 0.38
GSK3B P49841 3/20 0.38
DYRK1A Q13627 3/20 0.38
CLK2 P49760 1/20 0.38
CLK3 P49761 1/20 0.38
MELK Q14680 1/20 0.37
KDM4E B2RXH2 2/20 0.36
AVPR1B P47901 1/20 0.36
PDK1 Q15118 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
SMN1; SMN2 Q16637 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592632 0.96 CTSL (0.45) CTSLCTSBCTSSCTSKCYP2D6
SCHEMBL5592732 0.92 CTSL (0.45) CTSLCTSBCTSSCTSKWNT1
SCHEMBL5593180 0.92 CTSL (0.45) CTSLCTSBCTSSCTSKPTGER1
SCHEMBL5592691 0.91 CTSS (0.49) CTSLCTSBCTSSCTSKMELK
SCHEMBL5592898 0.90 CTSL (0.43) CTSLCTSBCTSSCTSKWNT1
SCHEMBL5592899 0.88 CHEK1 (0.38) CTSLCTSBCTSSCTSKKDM4E
Trifluoroacetic Acid SCHEMBL5592864 0.83 CTSS (0.47) CTSLCTSBCTSSCTSKCYP2C9
SCHEMBL5593161 0.82 CTSL (0.60) CTSLCTSBCTSSCTSKCYP2D6
Trifluoroacetic Acid SCHEMBL5592645 0.82 CTSS (0.47) CTSLCTSBCTSSCTSKMELK
SCHEMBL5592704 0.82 CTSS (0.59) CTSLCTSBCTSSCTSKMELK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed