SCHEMBL5592899

SCHEMBL5592899

CC(C)CNN(C(=O)c1cccc(CN2C(C)CCCC2C)c1)c1nc(C#N)ncc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.38
ACHE P22303 1/20 0.38
CTSL P07711 3/20 0.36
CTSS P25774 3/20 0.36
CTSK P43235 2/20 0.36
CTSB P07858 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
CHRM4 P08173 1/20 0.32
BRD4 O60885 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
CHRM2 P08172 1/20 0.32
CHRM1 P11229 1/20 0.32
ACKR3 P25106 1/20 0.31
HSD11B1 P28845 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592803 0.91 CTSS (0.41) CHEK1ACHECTSLCTSSCTSK
SCHEMBL5592852 0.88 CTSL (0.43) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL5592632 0.85 CTSL (0.45) CTSLCTSSCTSKCTSBKDM4E
SCHEMBL5593180 0.84 CTSL (0.45) ACHECTSLCTSSCTSKCTSB
SCHEMBL5592732 0.84 CTSL (0.45) ACHECTSLCTSSCTSKCTSB
SCHEMBL5593179 0.83 CTSL (0.51) CHEK1ACHECTSLCTSSCTSK
SCHEMBL5592898 0.82 CTSL (0.43) ACHECTSLCTSSCTSKCTSB
Trifluoroacetic Acid SCHEMBL5592740 0.79 CTSL (0.47) CHEK1ACHECTSLCTSSCTSK
SCHEMBL5592691 0.78 CTSS (0.49) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5592894 0.75 CTSL (0.45) CTSLCTSSCTSKCTSBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed