SCHEMBL5593246

SCHEMBL5593246

CC(C)CN(NC(=O)c1ccc(CN2CCC2)cc1)c1nc(C#N)ncc1Br

nearest known ligand 0.87

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.87
CTSS P25774 2/20 0.87
CTSK P43235 2/20 0.87
CTSB P07858 1/20 0.87
HDAC1 Q13547 5/20 0.40
HDAC6 Q9UBN7 3/20 0.40
HDAC8 Q9BY41 1/20 0.40
TBK1 Q9UHD2 2/20 0.37
CHRM2 P08172 1/20 0.36
PRKAA2 P54646 2/20 0.36
MELK Q14680 1/20 0.36
HDAC4 P56524 2/20 0.36
MCHR1 Q99705 1/20 0.35
PTGER1 P34995 2/20 0.35
KCNH2 Q12809 1/20 0.35
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5592618 0.98 CTSL (0.87) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5593209 0.97 CTSL (0.86) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5592896 0.93 CTSS (1.00) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL8245186 0.93 CTSL (0.83) CTSLCTSSCTSKCTSBALDH1A1
Trifluoroacetic Acid SCHEMBL5592621 0.92 CTSL (0.78) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5592822 0.92 CTSS (0.88) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL5592866 0.89 CTSL (0.72) CTSLCTSSCTSKCTSBHDAC1
Trifluoroacetic Acid SCHEMBL3319243 0.88 CTSS (0.90) CTSLCTSSCTSKCTSBHDAC6
SCHEMBL8242433 0.88 CTSL (0.71) CTSLCTSSCTSKCTSBHDAC1
SCHEMBL8245022 0.88 CTSS (0.85) CTSLCTSSCTSKCTSBHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO claimed
WO-2007025775-A2 CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2007-03-08 WO disclosed