SCHEMBL5597097

SCHEMBL5597097

CN(C)Cc1cccc(COc2n[c]c(-c3nc4ccccc4s3)cn2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
RAB9A P51151 4/20 0.38
MAPT P10636 3/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
NFKB1 P19838 2/20 0.38
NFKB2 Q00653 2/20 0.38
RELA Q04206 2/20 0.38
TDP1 Q9NUW8 1/20 0.38
CYP3A4 P08684 2/20 0.38
NOS1 P29475 2/20 0.37
NOS2 P35228 1/20 0.37
APP P05067 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.36
MGMT P16455 1/20 0.36
LCK P06239 1/20 0.36
ITK Q08881 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5596467 0.81 NPC1 (0.48) RAB9AMAPTSMN1; SMN2CYP3A4L3MBTL1
SCHEMBL4949283 0.80 ATP4A (0.41) RAB9AMAPTSMN1; SMN2NFKB1NFKB2
SCHEMBL4949209 0.79 ATP4A (0.45) RAB9AMAPTSMN1; SMN2NFKB1NFKB2
SCHEMBL5596393 0.77 KDM4E (0.36) PTGS1PTGS2RAB9AMAPTSMN1; SMN2
SCHEMBL5596344 0.76 RAB9A (0.46) RAB9AMAPTSMN1; SMN2NFKB1NFKB2
SCHEMBL4949763 0.73 MAPK8 (0.41) RAB9AMAPTSMN1; SMN2APPNPC1
SCHEMBL4948593 0.72 MAPK8 (0.55) PTGS1PTGS2RAB9AMAPTSMN1; SMN2
SCHEMBL4949279 0.72 MGLL (0.43) RAB9ASMN1; SMN2KDM4ENPC1TP53
SCHEMBL4947760 0.72 APP (0.41) RAB9AMAPTSMN1; SMN2NOS1APP
SCHEMBL2885027 0.69 MAPK10 (0.76) PTGS1PTGS2MAPTSMN1; SMN2TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1696909-B1 BENZOTHIAZOLE DERIVATIVES FOR THE TREATMENT OF DIABETES SERONO LAB (CH) 2007-11-14 EP claimed