SCHEMBL5599230

SCHEMBL5599230

O=C(N1CCCC1)N1c2ccc(F)cc2C2(CCNCC2)[C@H]1CC1CC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 5/20 0.38
TPSD1 Q9BZJ3 5/20 0.38
TPSG1 Q9NRR2 5/20 0.38
DPP4 P27487 1/20 0.36
SMYD3 Q9H7B4 3/20 0.36
CHRM2 P08172 1/20 0.34
CHRM3 P20309 1/20 0.34
KDM1A O60341 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP3A4 P08684 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRK1 P41145 1/20 0.34
OPRL1 P41146 1/20 0.34
CTSS P25774 2/20 0.33
USP2 O75604 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
GNRHR P30968 1/20 0.32
KCNH2 Q12809 1/20 0.32
NAMPT P43490 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5616077 0.99 TPSAB1 (0.38) TPSAB1TPSD1TPSG1DPP4SMYD3
SCHEMBL5599362 0.91 TPSAB1 (0.37) TPSAB1TPSD1TPSG1DPP4SMYD3
SCHEMBL5600486 0.85 GNRHR (0.36) TPSAB1TPSD1TPSG1DPP4SMYD3
SCHEMBL5599755 0.85 KDM1A (0.35) DPP4SMYD3KDM1AOPRM1OPRK1
SCHEMBL5599714 0.85 LMNA (0.36) DPP4KDM1AOPRM1OPRK1OPRL1
SCHEMBL5599739 0.84 OPRM1 (0.36) DPP4KDM1AALDH1A1OPRM1OPRK1
SCHEMBL5783985 0.84 DPP4 (0.34) DPP4KDM1AGNRHRKCNH2
SCHEMBL5782306 0.82 HTR2A (0.40) DPP4SMYD3KDM1ACYP2C19GNRHR
SCHEMBL5599501 0.82 KDM1A (0.37) DPP4KDM1AALDH1A1OPRM1OPRK1
SCHEMBL5599358 0.82 PARP1 (0.36) DPP4KDM1AGNRHRKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed