SCHEMBL5599362

SCHEMBL5599362

O=C(N1CCOCC1)N1c2ccc(F)cc2C2(CCNCC2)[C@H]1CC1CC1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
DPP4 P27487 1/20 0.36
AKR1C3 P42330 1/20 0.36
CTSS P25774 5/20 0.36
CTSL P07711 2/20 0.36
CTSK P43235 2/20 0.36
CNR1 P21554 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
PKM P14618 1/20 0.33
ALDH1A1 P00352 1/20 0.33
GABRA1 P14867 1/20 0.33
GABRA3 P34903 1/20 0.33
GABRB2 P47870 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5599230 0.91 TPSAB1 (0.38) TPSAB1TPSD1TPSG1DPP4CTSS
SCHEMBL5616077 0.90 TPSAB1 (0.38) TPSAB1TPSD1TPSG1DPP4CTSS
SCHEMBL5599427 0.86 DPP4 (0.36) DPP4AKR1C3CTSSCTSLCTSK
SCHEMBL5783985 0.82 DPP4 (0.34) DPP4
SCHEMBL5599755 0.81 KDM1A (0.35) DPP4MEN1KMT2ASMYD3
SCHEMBL5599714 0.81 LMNA (0.36) DPP4MEN1KMT2A
SCHEMBL5782306 0.80 HTR2A (0.40) DPP4SMYD3
SCHEMBL5599739 0.80 OPRM1 (0.36) DPP4CTSSMEN1KMT2AALDH1A1
SCHEMBL5599501 0.80 KDM1A (0.37) DPP4ALDH1A1
SCHEMBL5599358 0.80 PARP1 (0.36) DPP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed