SCHEMBL5599427

SCHEMBL5599427

C=CC[C@H]1N(C(=O)N2CCOCC2)c2ccc(F)cc2C12CCNCC2

nearest known ligand 0.36

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.36
AKR1C3 P42330 1/20 0.35
GNRHR P30968 1/20 0.35
PRKAG1 P54619 1/20 0.35
PRKAA1 Q13131 1/20 0.35
PRKAB1 Q9Y478 1/20 0.35
HDAC6 Q9UBN7 1/20 0.33
CNR1 P21554 1/20 0.33
ALDH1A1 P00352 2/20 0.33
KMT2A Q03164 2/20 0.33
MAPT P10636 1/20 0.33
PKM P14618 1/20 0.33
CTSS P25774 3/20 0.33
KIF11 P52732 1/20 0.33
CTSL P07711 1/20 0.32
CTSK P43235 1/20 0.32
FKBP1A P62942 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5600486 0.92 GNRHR (0.36) DPP4GNRHRALDH1A1KMT2AMEN1
SCHEMBL5599362 0.86 TPSAB1 (0.37) DPP4AKR1C3PRKAG1PRKAA1PRKAB1
SCHEMBL5786885 0.82 GNRHR (0.33) DPP4GNRHRCNR1KMT2AMEN1
SCHEMBL5778387 0.79 OPRM1 (0.35) DPP4GNRHR
SCHEMBL5599105 0.79 CHRNB2 (0.34) DPP4GNRHR
SCHEMBL5780824 0.79 GNRHR (0.37) DPP4GNRHRHDAC6
SCHEMBL5786887 0.77 GNRHR (0.41) GNRHR
SCHEMBL5599768 0.77 GNRHR (0.36) DPP4GNRHR
SCHEMBL5780422 0.77 P2RX7 (0.36) DPP4GNRHRALDH1A1
SCHEMBL5599230 0.77 TPSAB1 (0.38) DPP4GNRHRALDH1A1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005063745-A9 NOVEL SPIROINDOLINE OR SPIROISOQUINOLINE COMPOUNDS, METHODS OF USE AND COMPOSITIONS THEREOF ARENA PHARM INC (US) 2007-02-01 WO claimed