SCHEMBL5608905

SCHEMBL5608905

O=C1[N]Nc2cc(-c3ccccc3)c([N+](=O)[O-])cc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 1/20 0.40
STAT6 P42226 1/20 0.40
HIF1A Q16665 1/20 0.40
PHLPP2 Q6ZVD8 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MEN1 O00255 4/20 0.38
KMT2A Q03164 4/20 0.38
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PSMD14 O00487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15461976 0.79 ALDH1A1 (0.69) ALDH1A1TDP1CRHBPCRHR2TP53
SCHEMBL5608922 0.79 MAOA (0.40) ALDH1A1TP53CYP1A2CYP3A4CYP2D6
SCHEMBL5608736 0.76 TSHR (0.40) ALDH1A1CYP3A4MAPK1LMNA
SCHEMBL22007056 0.74 ALDH1A1 (0.67) ALDH1A1TDP1CRHBPCRHR2TP53
SCHEMBL5068702 0.70 ALDH1A1 (0.56) ALDH1A1TDP1CRHBPCRHR2TP53
SCHEMBL17742484 0.70 ALDH1A1 (0.60) ALDH1A1TDP1CRHBPCRHR2TP53
SCHEMBL23609775 0.69 ALDH1A1 (0.55) ALDH1A1TDP1CRHBPCRHR2TP53
SCHEMBL5259225 0.69 CAPN9 (0.54) ALDH1A1TDP1CYP3A4MEN1KMT2A
SCHEMBL6820729 0.69 PTPRC (0.50) ALDH1A1TDP1CYP1A2CYP3A4HIF1A
SCHEMBL17915595 0.68 ALDH1A1 (0.58) ALDH1A1TDP1CRHBPCRHR2TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797042-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2007-06-20 EP disclosed
WO-2006034804-A1 INDOZOLONE DERIVATIVES AS 11B-HSD1 INHIBITORS F.HOFFMANN-LA ROCHE AG (CH) 2006-04-06 WO disclosed