Predicted protein targets (top 20)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | MAPT | P10636 | 2/20 | 0.43 |
| ▸ | ALDH1A1 | P00352 | 2/20 | 0.43 |
| ▸ | PTGS1 | P23219 | 3/20 | 0.37 |
| ▸ | PTGS2 | P35354 | 3/20 | 0.37 |
| ▸ | MGLL | Q99685 | 2/20 | 0.37 |
| ▸ | TP53 | P04637 | 1/20 | 0.37 |
| ▸ | GAA | P10253 | 1/20 | 0.37 |
| ▸ | FAAH | O00519 | 1/20 | 0.37 |
| ▸ | KMT2A | Q03164 | 2/20 | 0.36 |
| ▸ | L3MBTL1 | Q9Y468 | 2/20 | 0.35 |
| ▸ | MEN1 | O00255 | 1/20 | 0.35 |
| ▸ | USP2 | O75604 | 1/20 | 0.35 |
| ▸ | CYP1A2 | P05177 | 1/20 | 0.35 |
| ▸ | POLB | P06746 | 1/20 | 0.35 |
| ▸ | CYP3A4 | P08684 | 1/20 | 0.35 |
| ▸ | THRB | P10828 | 1/20 | 0.35 |
| ▸ | CYP2C9 | P11712 | 1/20 | 0.35 |
| ▸ | HPGD | P15428 | 1/20 | 0.35 |
| ▸ | ALOX12 | P18054 | 1/20 | 0.35 |
| ▸ | CYP2C19 | P33261 | 1/20 | 0.35 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL5633937 | 0.83 | TDP1 (0.54) | MAPTALDH1A1MGLLFAAHKMT2A | |
| SCHEMBL5633265 | 0.83 | AGTR1 (0.40) | MAPTALDH1A1KMT2AL3MBTL1CYP1A2 | |
| SCHEMBL5633809 | 0.82 | TDP1 (0.56) | MAPTALDH1A1MGLLFAAHKMT2A | |
| SCHEMBL30943142 | 0.82 | ALDH1A1 (0.36) | MAPTALDH1A1SMN1; SMN2 | |
| SCHEMBL22212835 | 0.81 | ALDH1A1 (0.35) | MAPTALDH1A1PTGS1PTGS2MGLL | |
| SCHEMBL30943067 | 0.81 | TLR7 (0.35) | MAPTALDH1A1L3MBTL1 | |
| SCHEMBL5634058 | 0.81 | CDC25B (0.37) | MAPTALDH1A1L3MBTL1CYP2C9CYP2C19 | |
| SCHEMBL5633330 | 0.80 | CDC25B (0.38) | MAPTALDH1A1L3MBTL1CYP2C9HPGD | |
| SCHEMBL5633433 | 0.80 | CDC25B (0.38) | MAPTALDH1A1L3MBTL1CYP2C9HPGD | |
| SCHEMBL5634034 | 0.80 | CDC25B (0.38) | MAPTALDH1A1L3MBTL1CYP2C9HPGD |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20070123548-A1 | Pth agonists | COWAN DAVID J | 2007-05-31 | — | — | US | claimed |
| EP-1713782-A1 | PTH AGONISTS | SMITHKLINE BEECHAM CORPORATION (US) | 2006-10-25 | — | — | EP | claimed |
| WO-2005077918-A1 | PTH AGONISTS | SMITHKLINE BEECHAM CORPORATION (US) | 2005-08-25 | — | — | WO | claimed |
| US-11001820-B2 | Delivery of therapeutic agents by a collagen binding protein | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2021-05-11 | — | — | US | disclosed |
| US-20190249163-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSA S (US) | 2019-08-15 | — | — | US | disclosed |
| US-10358471-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2019-07-23 | — | — | US | disclosed |
| US-20190135890-A1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2019-05-09 | — | — | US | disclosed |
| US-10202434-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2019-02-12 | — | — | US | disclosed |
| EP-3091075-B1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | UNIV ARKANSAS (US) | 2018-06-13 | — | — | EP | disclosed |
| US-20170204390-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2017-07-20 | — | — | US | disclosed |
| US-20170204390-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2017-07-20 | — | — | US | disclosed |
| US-20150038423-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT | 2015-02-05 | — | — | US | disclosed |
| US-20140377215-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSA (US) | 2014-12-25 | — | — | US | disclosed |
| US-20140377215-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSA (US) | 2014-12-25 | — | — | US | disclosed |
| US-8450273-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2013-05-28 | — | — | US | disclosed |
| US-8450273-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2013-05-28 | — | — | US | disclosed |
| US-20100129341-A1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | OCHSNER CLINIC FOUNDATION | 2010-05-27 | — | — | US | disclosed |
| US-20100129341-A1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | OCHSNER CLINIC FOUNDATION | 2010-05-27 | — | — | US | disclosed |
| WO-2008124166-A2 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | THE BOARD OF TRUSTEES OF THE UNIVERSITY OF ARKANSAS (US) | 2008-10-16 | — | — | WO | disclosed |
| US-20070123548-A1 | Pth agonists | COWAN DAVID J | 2007-05-31 | — | — | US | disclosed |
Patent text — is the patent's own abstract consistent with the prediction?
For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.
| Patent | Title | Text reads most about | Predicted target · text-rank |
|---|---|---|---|
| US-20100129341-A1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | PTH1R, CALCRL, CALCR | MAPT 2450/4885ALDH1A1 4476/4885PTGS1 3311/4885 |
| US-10358471-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | PTH1R, CALCRL, CALCR | MAPT 2450/4885ALDH1A1 4476/4885PTGS1 3311/4885 |
| US-20170204390-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | PTH1R, GHRHR, FGF23 | MAPT 792/4885ALDH1A1 4687/4885PTGS1 3549/4885 |
| US-20070123548-A1 | Pth agonists | PTH1R, SSTR3, CALCR | MAPT 4835/4885ALDH1A1 3899/4885PTGS1 2325/4885 |
| US-20190135890-A1 | FUSION PROTEINS OF COLLAGEN-BINDING DOMAIN AND PARATHYROID HORMONE | PTH1R, CALCRL, CALCR | MAPT 2450/4885ALDH1A1 4476/4885PTGS1 3311/4885 |
| US-20150038423-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | PTH1R, CALCRL, CALCR | MAPT 1947/4885ALDH1A1 4586/4885PTGS1 2855/4885 |
| US-10202434-B2 | Fusion proteins of collagen-binding domain and parathyroid hormone | PTH1R, CALCRL, CALCR | MAPT 2450/4885ALDH1A1 4476/4885PTGS1 3311/4885 |
| US-20140377215-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | PTH1R, GHRHR, FGF23 | MAPT 792/4885ALDH1A1 4687/4885PTGS1 3549/4885 |
| US-11001820-B2 | Delivery of therapeutic agents by a collagen binding protein | PTH1R, GHRHR, FGF23 | MAPT 792/4885ALDH1A1 4687/4885PTGS1 3549/4885 |
| US-20190249163-A1 | DELIVERY OF THERAPEUTIC AGENTS BY A COLLAGEN BINDING PROTEIN | PTH1R, GHRHR, FGF23 | MAPT 792/4885ALDH1A1 4687/4885PTGS1 3549/4885 |
“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.