SCHEMBL5636028

SCHEMBL5636028

CC(C)(C)OC(=O)N1CCC(c2n[nH]c(Cc3ccccc3)n2)CC1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.51
GAA P10253 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
STS P08842 1/20 0.48
LMNA P02545 1/20 0.48
GPR119 Q8TDV5 4/20 0.47
TP53 P04637 2/20 0.47
PRMT5 O14744 2/20 0.47
MAPT P10636 1/20 0.47
TDP1 Q9NUW8 1/20 0.47
HPGDS O60760 1/20 0.46
KDM4E B2RXH2 1/20 0.46
PKM P14618 1/20 0.46
ACHE P22303 1/20 0.46
HTT P42858 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14539183 0.84 RIPK1 (0.41)
SCHEMBL4343857 0.81 HPGDS (0.55) THRBGAASMN1; SMN2STSLMNA
SCHEMBL5763660 0.80 HTT (0.58) THRBGAASMN1; SMN2STSLMNA
SCHEMBL5763947 0.79 HPGDS (0.53) THRBGAASMN1; SMN2STSLMNA
SCHEMBL29024490 0.79 DRD2 (0.59) THRBGAASMN1; SMN2STSLMNA
SCHEMBL14514120 0.79 THRB (0.51) THRBGAASMN1; SMN2STSLMNA
SCHEMBL29024484 0.79 THRB (0.52) THRBGAASMN1; SMN2STSLMNA
SCHEMBL1137864 0.76 GPR119 (0.53) THRBGPR119PRMT5MAPTHPGDS
SCHEMBL14829908 0.76 KDM4E (0.49) THRBGPR119MAPTKDM4EHTT
SCHEMBL15878935 0.76 MAPT (0.49) THRBGPR119MAPTHPGDSKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed
US-7217714-B1 CCR5 modulators AGOURON PHARMACEUTICALS, INC. (US) 2007-05-15 US disclosed