SCHEMBL5639142

SCHEMBL5639142

O=C1O[C@@H](CO)CN1c1ccc(-c2ccon2)cc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CALML3 P27482 6/20 0.51
MAOA P21397 3/20 0.49
MAOB P27338 3/20 0.49
GRM2 Q14416 4/20 0.42
CYP2C19 P33261 2/20 0.42
CYP2C9 P11712 1/20 0.42
CYP3A4 P08684 1/20 0.41
P2RX3 P56373 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14603044 0.88 F10 (0.53) CALML3MAOAGRM2
SCHEMBL6271162 0.81 GRM2 (0.38) GRM2P2RX3
SCHEMBL5637293 0.81 GRM2 (0.42) GRM2
SCHEMBL9550251 0.79 MAOA (0.59) CALML3MAOAMAOBGRM2
SCHEMBL5637317 0.78 MAOA (0.57) MAOAGRM2
SCHEMBL9549439 0.77 GRM2 (0.64) CALML3MAOAMAOBGRM2
SCHEMBL9482302 0.77 GRM2 (0.64) CALML3MAOAMAOBGRM2
SCHEMBL6606264 0.76 ITGB3 (0.58) CALML3MAOAMAOBGRM2
SCHEMBL3323919 0.76 MAOA (0.58) CALML3MAOAMAOBGRM2
SCHEMBL7297166 0.76 GRM2 (0.63) CALML3MAOAMAOBGRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7157482-B2 Antibacterial 1,3-oxazolidin-2-one derivatives ASTRAZENECA AB (SE) 2007-01-02 US disclosed
US-20060084810-A1 Antibacterial 1,3-oxazolidin-2-one derivatives ASTRAZENECA AB (SE) 2006-04-20 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060084810-A1 Antibacterial 1,3-oxazolidin-2-one derivatives HRH1, HDHD5, NGLY1 CALML3 4277/4885MAOA 717/4885MAOB 898/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.