SCHEMBL5644297

SCHEMBL5644297

C=C(COCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 18/20 0.52
CACNA1F O60840 3/20 0.52
CACNA1D Q01668 3/20 0.52
CACNA1S Q13698 3/20 0.52
CACNA1C Q13936 3/20 0.52
SLC6A4 P31645 3/20 0.45
IDO1 P14902 1/20 0.44
P2RX1 P51575 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1872900 0.85 TACR1 (0.52) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL21596609 0.79 TSHR (0.54) IDO1
SCHEMBL8621299 0.77 ALDH1A1 (0.42)
SCHEMBL7496743 0.74 IDO1 (0.52) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL13307223 0.74 TACR1 (0.58) TACR1
SCHEMBL8963934 0.73 TACR1 (0.59) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL3752087 0.73 MAOA (0.50)
SCHEMBL1873597 0.72 PLOD2 (0.46) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL8880647 0.72 TACR1 (0.48) TACR1CACNA1FCACNA1DCACNA1SCACNA1C
SCHEMBL27591269 0.72 MAOA (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7179926-B2 Aryloxyalkylamine NK-1/SSRI inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-02-20 US disclosed
WO-2006014942-A1 ARYLOXYALKYLAMINE NK-1/SSRI INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2006-02-09 WO disclosed
US-20060020019-A1 Aryloxyalkylamine NK-1/SSRI inhibitors BRISTOL-MYERS SQUIBB COMPANY 2006-01-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060020019-A1 Aryloxyalkylamine NK-1/SSRI inhibitors TPH1, SLC6A4, HTR1A TACR1 26/4885CACNA1F 704/4885CACNA1D 549/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.