SCHEMBL5644659

SCHEMBL5644659

FC(F)(F)COc1ccc(Cl)nn1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.44
CHRNB2 P17787 1/20 0.41
CHRNA4 P43681 1/20 0.41
MAPT P10636 3/20 0.40
CYP1A2 P05177 1/20 0.38
ALDH1A1 P00352 2/20 0.37
RECQL P46063 1/20 0.37
IL1B P01584 1/20 0.36
EPHX2 P34913 1/20 0.36
GAA P10253 1/20 0.35
POLB P06746 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4949662 0.78 CHRNA4 (0.39) SMN1; SMN2CHRNB2CHRNA4MAPTALDH1A1
SCHEMBL22655057 0.78 IL1B (0.46) SMN1; SMN2CHRNB2CHRNA4MAPTALDH1A1
SCHEMBL23148685 0.77 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL28670107 0.77 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL29637301 0.77 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL29685778 0.77 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL16705085 0.77 SMN1; SMN2 (0.49) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL19664476 0.76 SMN1; SMN2 (0.48) SMN1; SMN2L3MBTL1MAPTCYP1A2ALDH1A1
SCHEMBL3063761 0.74 CHRNB2 (0.42) CHRNB2CHRNA4MAPTALDH1A1GAA
SCHEMBL2492398 0.74 HTT (0.45) SMN1; SMN2CHRNB2CHRNA4MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2026-04-16 US disclosed
US-12435083-B2 Cyclopropyl-(hetero)aryl-substituted ethylsulphonyl-pyridine derivatives BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2025-10-07 US disclosed
CN-118355004-A Cyclopropyl- (heteroaryl) -substituted ethylsulfonyl-pyridine derivatives 勃林格殷格翰动物保健有限公司 2024-07-16 CN disclosed
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2023-07-27 US disclosed
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2023-07-27 US disclosed
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2023-07-27 US disclosed
WO-2023036934-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYLPYRIDINE DERIVATIVES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2023-03-16 WO disclosed
US-7179806-B2 Δ1-pyrrolines used as pesticides BAYER CROPSCIENCE AG (DE) 2007-02-20 US disclosed
US-7179806-B2 Δ1-pyrrolines used as pesticides BAYER CROPSCIENCE AG (DE) 2007-02-20 US disclosed
US-7179806-B2 Δ1-pyrrolines used as pesticides BAYER CROPSCIENCE AG (DE) 2007-02-20 US disclosed
EP-1347957-B1 DELTA 1-PYRROLINES USED AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2005-09-07 EP disclosed
US-20040082586-A1 Delta 1-pyrrolines used as pesticides BAYER CROPSCIENCE AG (DE) 2004-04-29 US disclosed
EP-1347957-A1 DELTA 1-PYRROLINES USED AS PESTICIDES Bayer CropScience AG (DE) 2003-10-01 EP disclosed
WO-2002046151-A1 DELTA 1-PYRROLINES USED AS PESTICIDES BAYER CROPSCIENCE AG (DE) 2002-06-13 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES CYCS, CYP2E1, AHR SMN1; SMN2 4334/4885L3MBTL1 2181/4885CHRNB2 3006/4885
US-12435083-B2 Cyclopropyl-(hetero)aryl-substituted ethylsulphonyl-pyridine derivatives CYCS, CYP2E1, CYP1A1 SMN1; SMN2 4257/4885L3MBTL1 1985/4885CHRNB2 3027/4885
US-20040082586-A1 Delta 1-pyrrolines used as pesticides DDT, CHRM1, PRMT1 SMN1; SMN2 1915/4885L3MBTL1 572/4885CHRNB2 447/4885
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES CBR3, CYCS, CBR1 SMN1; SMN2 3977/4885L3MBTL1 211/4885CHRNB2 1329/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.