SCHEMBL5657166

SCHEMBL5657166

COCNC(=O)COc1ncc(C(=O)O)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 6/20 0.40
KDM4E B2RXH2 2/20 0.38
HSD17B10 Q99714 2/20 0.38
ALDH1A1 P00352 1/20 0.38
ALOX15 P16050 1/20 0.38
CSNK2A2 P19784 1/20 0.36
CSNK2A1 P68400 1/20 0.36
MAPT P10636 1/20 0.36
MAPK1 P28482 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
XDH P47989 1/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
USP2 O75604 1/20 0.34
HCAR2 Q8TDS4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5658255 0.77 KMT2A (0.61) KDM4EALDH1A1MAPTL3MBTL1CYP1A2
SCHEMBL15514113 0.74 HCAR3 (0.50) HCAR3KDM4EHSD17B10ALDH1A1ALOX15
SCHEMBL5660811 0.73 GAA (0.60) KDM4EALDH1A1MAPTMAPK1L3MBTL1
SCHEMBL5658844 0.73 CXCR1 (0.53) KDM4EALDH1A1L3MBTL1SMN1; SMN2MEN1
SCHEMBL5660559 0.72 MAPT (0.45) HCAR3KDM4EHSD17B10ALDH1A1ALOX15
SCHEMBL5658335 0.71 KDM4E (0.50) HCAR3KDM4EHSD17B10ALDH1A1ALOX15
SCHEMBL186124 0.71 MAPT (0.59) HCAR3KDM4EHSD17B10ALDH1A1ALOX15
SCHEMBL5657170 0.71 KDM4E (0.46) HCAR3KDM4EHSD17B10ALDH1A1ALOX15
SCHEMBL5659943 0.71 KMT2A (0.52) HCAR3HSD17B10ALDH1A1MAPK1L3MBTL1
SCHEMBL5660210 0.71 SMN1; SMN2 (0.55) KDM4EALDH1A1MAPTL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7176310-B1 Pyrimidinecarboxamide derivatives and their use as anti-inflammatory agents UCB SA (GB) 2007-02-13 US disclosed