SCHEMBL567474

SCHEMBL567474

COc1cccc2c1C(=O)c1c(O)c3c(c(O)c1C2=O)CC(O)CC3

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.54
PIM1 P11309 1/20 0.54
ELANE P08246 8/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
CTSG P08311 1/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
TCF4 P15884 1/20 0.43
CTNNB1 P35222 1/20 0.43
ELAVL1 Q15717 1/20 0.43
MAPT P10636 2/20 0.42
RAB9A P51151 2/20 0.42
POLL Q9UGP5 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
S100A4 P26447 1/20 0.42
NPC1 O15118 1/20 0.42
SOS1 Q07889 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14537729 1.00 EGFR (0.54) EGFRPIM1ELANEMEN1KMT2A
Hydrochloric Acid SCHEMBL7460 0.99 EGFR (0.53) EGFRPIM1ELANEMEN1KMT2A
Hydrochloric Acid SCHEMBL29658548 0.99 EGFR (0.53) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL13452107 0.87 EGFR (0.53) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL17278322 0.86 EGFR (0.52) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL21573136 0.86 EGFR (0.52) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL21886965 0.85 EGFR (0.51) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL22873368 0.85 EGFR (0.51) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL11395596 0.85 EGFR (0.51) EGFRPIM1ELANEMEN1KMT2A
SCHEMBL11429902 0.85 EGFR (0.51) EGFRPIM1ELANEMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0007403-B1 5,12-DIHYDROXY-1,2,3,4,6,11-HEXAHYDRO-2,6,11-TRIOXONAPHTHACENES AND THEIR SYNTHESIS THE UNIVERSITY OF KANSAS (US) 1982-11-24 EP claimed
US-4244880-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1981-01-13 US claimed
US-4215062-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1980-07-29 US claimed
EP-0007403-A1 5,12-dihydroxy-1,2,3,4,6,11-hexahydro-2,6,11-trioxonaphthacenes and their synthesis THE UNIVERSITY OF KANSAS (US) 1980-02-06 EP claimed
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY ZOUNEK ALEX (DE) 2025-12-18 US disclosed
US-20240239764-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2024-07-18 US disclosed
US-20240083868-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS MEKANISTIC THERAPEUTICS, LLC 2024-03-14 US disclosed
US-20240050415-A1 DACLATASVIR FOR USE IN TREATING LUNG AND PROSTATE CANCER HENRY FORD HEALTH SYSTEM (US) 2024-02-15 US disclosed
US-11673876-B2 Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors MEKANISTIC THERAPEUTICS LLC (US) 2023-06-13 US disclosed
WO-2023078273-A1 SPECIFIC CONJUGATION FOR AN ANTIBODY-DRUG CONJUGATE HANGZHOU DAC BIOTECH CO., LTD. (CN) 2023-05-11 WO disclosed
US-20220213054-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS MEKANISTIC THERAPEUTICS LLC (US) 2022-07-07 US disclosed
US-11141459-B2 Pharmaceutical composition comprising Lefty GRANT LABS, INC. (US) 2021-10-12 US disclosed
US-20090175869-A1 Pulsatile Dosing of Gossypol for Treatment of Disease ASCENTA THERAPEUTICS, INC. (US) 2009-07-09 US disclosed
US-20090010878-A1 Pulsatile dosing of gossypol for treatment of disease ASCENTA THERAPEUTICS, INC. (US) 2009-01-08 US disclosed
US-20080021095-A1 Small Molecule Antagonists of Xiap Family Proteins THE REGENTS OF THE UNIVERSITY OF MICHIGAN 2008-01-24 US disclosed
US-20050261232-A1 Non-natural ribonuclease conjugates as cytotoxic agents QUINTESSENCE BIOSCIENCES, INC. (US) 2005-11-24 US disclosed
EP-0007403-B1 5,12-DIHYDROXY-1,2,3,4,6,11-HEXAHYDRO-2,6,11-TRIOXONAPHTHACENES AND THEIR SYNTHESIS THE UNIVERSITY OF KANSAS (US) 1982-11-24 EP disclosed
US-4244880-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1981-01-13 US disclosed
US-4215062-A Anthracycline synthesis UNIVERSITY OF KANSAS ENDOWMENT ASSOCIATION (US) 1980-07-29 US disclosed
EP-0007403-A1 5,12-dihydroxy-1,2,3,4,6,11-hexahydro-2,6,11-trioxonaphthacenes and their synthesis THE UNIVERSITY OF KANSAS (US) 1980-02-06 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250381202-A1 PRODRUG KIT FOR MULTI-PRONGED CHEMOTHERAPY KIT, CTSL, PAICS EGFR 358/4885PIM1 961/4885ELANE 2347/4885
US-20240239764-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS EGFR, ERBB2, ERBB3 EGFR 1/4885PIM1 305/4885ELANE 2275/4885
US-11673876-B2 Substituted aminobenzyl heteroaryl compounds as EGFR and/or PI3K inhibitors EGFR, ERBB2, ERBB3 EGFR 1/4885PIM1 305/4885ELANE 2275/4885
US-20090010878-A1 Pulsatile dosing of gossypol for treatment of disease BCL2, BAX, PHLPP2 EGFR 4322/4885PIM1 1373/4885ELANE 2794/4885
US-20220213054-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS EGFR, ERBB2, ERBB3 EGFR 1/4885PIM1 305/4885ELANE 2275/4885
US-20090175869-A1 Pulsatile Dosing of Gossypol for Treatment of Disease BCL2, BAX, BAD EGFR 4411/4885PIM1 1182/4885ELANE 3427/4885
US-20240083868-A1 SUBSTITUTED AMINOBENZYL HETEROARYL COMPOUNDS AS EGFR AND/OR PI3K INHIBITORS EGFR, ERBB2, ERBB3 EGFR 1/4885PIM1 305/4885ELANE 2275/4885
US-20080021095-A1 Small Molecule Antagonists of Xiap Family Proteins XIAP, BIRC5, BIRC3 EGFR 4170/4885PIM1 2139/4885ELANE 484/4885
US-20050261232-A1 Non-natural ribonuclease conjugates as cytotoxic agents RNASE1, RNASEL, RNASEH1 EGFR 2869/4885PIM1 2913/4885ELANE 608/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.