SCHEMBL5690242

SCHEMBL5690242

Cc1cccnc1Cc1ccc(OC(=O)N2CCC(Sc3nnnn3CCN(C)C)CC2)cc1

nearest known ligand 0.36

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SMO Q99835 1/20 0.36
GRIN2B Q13224 4/20 0.35
DCUN1D1 Q96GG9 5/20 0.33
UBE2M P61081 4/20 0.33
GAA P10253 1/20 0.32
SSTR4 P31391 1/20 0.32
NPY2R P49146 1/20 0.32
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
KMT2A Q03164 1/20 0.31
TRPA1 O75762 2/20 0.31
TRPV1 Q8NER1 1/20 0.31
GCK P35557 1/20 0.31
KDM1A O60341 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5688420 0.93 GRIN2B (0.35) GRIN2BDCUN1D1UBE2MGAASSTR4
SCHEMBL5690035 0.91 SMO (0.38) SMOGRIN2BGAASSTR4NPY2R
SCHEMBL5688853 0.89 SMO (0.39) SMOGRIN2BGAANPY2RKMT2A
SCHEMBL5687343 0.89 SMO (0.39) SMOGRIN2BGAASSTR4NPY2R
SCHEMBL5687424 0.88 GAA (0.35) SMOGRIN2BDCUN1D1UBE2MGAA
SCHEMBL5688888 0.85 NOS3 (0.34) SMOGRIN2BDCUN1D1UBE2MKDM1A
SCHEMBL5688077 0.84 GAA (0.33) SMOGAASSTR4NPY2RALDH1A1
SCHEMBL5687632 0.84 UBE2M (0.36) SMODCUN1D1UBE2MGAAALDH1A1
SCHEMBL5688602 0.84 GRIN2B (0.34) SMOGRIN2BDCUN1D1UBE2MTRPV1
SCHEMBL5687919 0.83 LIPE (0.41) DCUN1D1UBE2MTRPA1TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20060160851-A1 Substituted piperidine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US claimed
EP-1636207-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2006-03-22 EP claimed
WO-2004111032-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2004-12-23 WO claimed
US-20060160851-A1 Substituted piperidine carbamates NOVO NORDISK A/S (DK) 2006-07-20 US disclosed
EP-1636207-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2006-03-22 EP disclosed
WO-2004111032-A1 SUBSTITUTED PIPERIDINE CARBAMATES FOR USE AS INHIBITORS OF HORMONE SENSITIVE LIPASE NOVO NORDISK A/S (DK) 2004-12-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060160851-A1 Substituted piperidine carbamates LIPE, PNLIP, LIPC SMO 3195/4885GRIN2B 2588/4885DCUN1D1 4035/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.