SCHEMBL570053

SCHEMBL570053

Cc1c(C(=O)O)n[nH]c1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 10/20 0.50
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4185273 0.80 ALOX15 (0.44) HCAR2KMT2A
SCHEMBL15825699 0.73 HCAR2 (0.58) HCAR2
SCHEMBL12985499 0.73 PDE4D (0.38) HCAR2KMT2A
SCHEMBL4631308 0.73 HCAR2 (0.63) HCAR2
SCHEMBL9912568 0.72 ABCC8 (0.54) HCAR2
SCHEMBL7234538 0.71 HCAR2 (0.57) HCAR2KMT2A
SCHEMBL1829755 0.71 L3MBTL1 (0.32) KMT2A
SCHEMBL12121211 0.70 DYRK1A (0.46)
SCHEMBL12263262 0.69 HCAR2 (0.55) HCAR2KMT2A
SCHEMBL31741716 0.69 HCAR2 (0.59) HCAR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3016934-A2 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME Millennium Pharmaceuticals, Inc. (US) 2016-05-11 EP disclosed
WO-2015002994-A2 HETEROARYL COMPOUNDS USEFUL AS INHIBITORS OF SUMO ACTIVATING ENZYME MILLENNIUM PHARMACEUTICALS, INC. (US) 2015-01-08 WO disclosed
EP-2601208-A2 LIGANDS FOR ANTIBODY AND Fc-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMATOGRAPHY Graffinity Pharmaceuticals GmbH (DE) 2013-06-12 EP disclosed
WO-2012017021-A2 LIGANDS FOR ANTIBODY AND Fc-FUSION PROTEIN PURIFICATION BY AFFINITY CHROMATOGRAPHY GRAFFINITY PHARMACEUTICALS GMBH (DE) 2012-02-09 WO disclosed