Bromfenac

Bromfenac

SCHEMBL57092

Nc1c(CC(=O)O)cccc1C(=O)c1ccc(Br)cc1.[Na]

nearest known ligand 0.97

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

PTGS1PTGS2

The experimentally established mechanism targets of Bromfenac. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS1 known ✓ P23219 1/20 0.97
PTGS2 known ✓ P35354 1/20 0.97
ABCB11 O95342 1/20 0.97
LMNA P02545 1/20 0.97
ADORA1 P30542 1/20 0.97
AKR1C3 P42330 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromfenac SCHEMBL34411 0.99 ABCB11 (1.00) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL14861906 0.99 ABCB11 (1.00) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL28429415 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL28895435 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL28429368 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL28429917 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL57090 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL4603047 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL28420990 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2
Bromfenac SCHEMBL15968905 0.97 ABCB11 (0.97) ABCB11LMNAPTGS1ADORA1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1905 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4615506-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES Sahin, Fikret (TR) 2025-09-17 EP claimed
US-20250281395-A1 OPHTHALMIC PREPARATION FOR TREATING MACULAR EDEMA, OPTIC NEURITIS AND NON-INFECTIOUS ENDOPHTHALMITIS THROUGH EYE DROP ADMINISTRATION Chengdu Ruimu Biopharmaceuticals Co., Ltd. (CN) 2025-09-11 US claimed
WO-2025081182-A1 CITRATE-BASED OCULAR IMPLANTS AND POLYMERS THE PENN STATE RESEARCH FOUNDATION (US) 2025-04-17 WO claimed
WO-2024258363-A1 USE OF GSK-3 ACTIVATIOR TO MODULATE PROTEASOME ACTIVITY TO PREVENT AGEING ASSOCIATED CONDITIONS AND DISEASES SAHIN FIKRET (TR) 2024-12-19 WO claimed
CN-118615245-A Sodium bromfenac eye drops and preparation method thereof 武汉五景药业有限公司 2024-09-10 CN claimed
US-20240282425-A1 AUTHENTICATION METHODS AND SYSTEMS FOR DISPENSED PRESCRIPTIONS LOW GORDON KEITH (US) 2024-08-22 US claimed
US-20240252429-A1 EXTENDED-WEAR SILICONE HYDROGEL CONTACT LENSES AND USES THEREOF OCUMEDIC, INC. 2024-08-01 US claimed
CN-118319894-A Pharmaceutical composition and application thereof 广州润尔眼科生物科技有限公司 2024-07-12 CN claimed
CN-113698308-B Synthesis method of bromfenac sodium 山东辰龙药业有限公司 2024-06-21 CN claimed
CN-118121709-A Ophthalmic pharmaceutical composition, and preparation method and application thereof 山东序列生物科技有限公司 2024-06-04 CN claimed
EP-1681065-A1 WATER-BASED COMPOSITION UNDERGOING REVERSIBLE THERMOGELATION Wakamoto Pharmaceutical Co., Ltd. (JP) 2006-07-19 EP claimed
WO-2005048979-A2 PHARMACEUTICAL COMPOSITION HAVING CASING WITH MULTIPLE MICRO TABLETS TORRENT PHARMACEUTICALS LIMITED (IN) 2005-06-02 WO claimed
EP-1443969-A2 NON-INCLUSION CYCLODEXTRIN COMPLEXES Decode Genetics EHF (IS) 2004-08-11 EP claimed
US-20030138399-A1 Anti-inflammatory therapy for inflammatory mediated infection REGENTS OF THE UNIVERSITY OF CALIFORNIA, THE 2003-07-24 US claimed
US-20030109492-A1 Non-inclusion cyclodextrin complexes DECODE GENETICS EHF. (IS) 2003-06-12 US claimed
WO-2003033025-A2 CYCLODEXTRIN COMPLEXES DECODE GENETICS EHF (IS) 2003-04-24 WO claimed
JP-2002544210-A 2002-12-24 JP claimed
CN-1353573-A Anti-inflammatory therapy for inflammatory mediated infection UNIV CALIFORNIA (US) 2002-06-12 CN claimed
EP-1202620-A1 ANTI-INFLAMMATORY THERAPY FOR INFLAMMATORY MEDIATED INFECTION The Regents of the University of California (US) 2002-05-08 EP claimed
WO-2000069255-A1 ANTI-INFLAMMATORY THERAPY FOR INFLAMMATORY MEDIATED INFECTION THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2000-11-23 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030109492-A1 Non-inclusion cyclodextrin complexes SI, CNDP2, NONO PTGS1 3863/4885PTGS2 4282/4885ABCB11 857/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.