SCHEMBL5712367

SCHEMBL5712367

CCn1c(SC)nc2ccc(I)cc2c1=O

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPK1 P28482 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
RAB9A P51151 1/20 0.45
DHFR P00374 6/20 0.45
MAPT P10636 3/20 0.43
KDM4E B2RXH2 2/20 0.43
LMNA P02545 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
TSHR P16473 2/20 0.42
ATM Q13315 1/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7100456 0.89 DHFR (0.43) ALDH1A1SMN1; SMN2DHFRKDM4ELMNA
SCHEMBL8401780 0.88 DHFR (0.43) ALDH1A1SMN1; SMN2DHFRKDM4ELMNA
SCHEMBL8401779 0.87 DHFR (0.42) ALDH1A1SMN1; SMN2DHFRKDM4ELMNA
SCHEMBL5712366 0.80 KDM4E (0.40) ALDH1A1MAPK1SMN1; SMN2KDM4ELMNA
SCHEMBL5712377 0.77 ALDH1A1 (0.52) ALDH1A1MAPK1SMN1; SMN2MAPTKDM4E
SCHEMBL5712356 0.75 MAPK1 (0.45) ALDH1A1MAPK1SMN1; SMN2MAPTKDM4E
SCHEMBL7887739 0.73 PDE7A (0.53) ALDH1A1DHFR
SCHEMBL7101435 0.72 ADORA2B (0.41) ALDH1A1SMN1; SMN2RAB9AKDM4EMEN1
SCHEMBL11675393 0.71 CA12 (0.54) ALDH1A1SMN1; SMN2DHFRKDM4E
SCHEMBL8424278 0.70 LMNA (0.43) ALDH1A1SMN1; SMN2RAB9AKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1344775-B1 Preparation of fungicidal quinazolinones and useful intermediates DU PONT (US) 2006-11-29 EP disclosed
EP-0922037-B1 PREPARATION OF FUNGICIDAL QUINAZOLINONES AND USEFUL INTERMEDIATES DU PONT (US) 2003-10-01 EP disclosed
EP-1344775-A1 Preparation of fungicidal quinazolinones and useful intermediates E.I. DU PONT DE NEMOURS AND COMPANY (US) 2003-09-17 EP disclosed