Levoleucovorin

Levoleucovorin

SCHEMBL571901

Nc1nc(=O)c2c([nH]1)NC[C@H](CNc1ccc(C(=O)N[C@@H](CCC(=O)O)C(=O)O)cc1)N2C=O

nearest known ligand 0.80

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHFR P00374 2/20 0.80
LMNA P02545 1/20 0.62
MTHFD1 P11586 3/20 0.58
SOST Q9BQB4 1/20 0.57
MTHFD2 P13995 3/20 0.51
FPGS Q05932 2/20 0.51
ATIC P31939 2/20 0.51
TYMS P04818 2/20 0.48
KDM4E B2RXH2 1/20 0.48
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
POLB P06746 1/20 0.48
GAA P10253 1/20 0.48
AKR1B1 P15121 1/20 0.48
HPGD P15428 1/20 0.48
TSHR P16473 1/20 0.48
PTGS2 P35354 1/20 0.48
KMT2A Q03164 1/20 0.48
HSD17B10 Q99714 1/20 0.48
TDP1 Q9NUW8 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Leucovorin SCHEMBL5132046 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Folinic Acid SCHEMBL29369091 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL21632556 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL4708750 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL8349 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL8350 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL571902 1.00 DHFR (0.80) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL9054117 0.99 DHFR (0.78) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL16207660 0.99 DHFR (0.78) DHFRLMNAMTHFD1SOSTMTHFD2
Leucovorin SCHEMBL9054183 0.99 DHFR (0.78) DHFRLMNAMTHFD1SOSTMTHFD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 377 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260124144-A1 COMPOSITIONS COMPRISING DISODIUM LEVOFOLINATE Acrotech Biopharma Inc. (US) 2026-05-07 US claimed
US-12564556-B1 Compositions comprising disodium levofolinate Acrotech Biopharma Inc. (US) 2026-03-03 US claimed
US-12539276-B1 Compositions comprising disodium levofolinate Acrotech Biopharma Inc. (US) 2026-02-03 US claimed
US-20250215039-A1 NUCLEOSIDES FOR TREATING CANCER PRIMEFOUR THERAPEUTICS INC (US) 2025-07-03 US claimed
WO-2025111482-A1 COMPLEXING AGENT SALT FORMULATIONS OF PHARMACEUTICAL COMPOUNDS AT LOW STOICHIOMETRIC RATIOS BEXSON BIOMEDICAL, INC. (US) 2025-05-30 WO claimed
WO-2025101623-A1 METHODS OF TREATING CANCER AMGEN INC. (US) 2025-05-15 WO claimed
WO-2025100428-A1 COMBINATION OF ANTI-CD147 ANTIBODY AND ANOTHER ANTITUMOR AGENT 第一三共株式会社 2025-05-15 WO claimed
US-20250127782-A1 METHODS OF TREATING CANCER AMGEN INC. 2025-04-24 US claimed
EP-3893913-B1 TRANSFERRIN RECEPTOR TARGETING PEPTIDES FRED HUTCHINSON CANCER CENTER (US) 2025-03-26 EP claimed
CN-119548521-A Anti-aging composition for middle-aged and elderly people 深圳奥萨制药有限公司 2025-03-04 CN claimed
CN-112691107-B Pharmaceutical composition and application thereof 北京斯利安药业有限公司 2022-09-02 CN claimed
US-20220211657-A1 METHODS OF TREATING GASTROINTESTINAL CANCERS AND TUMORS THEREOF USING COMBINATION THERAPY GEORGETOWN UNIVERSITY 2022-07-07 US claimed
EP-3099816-B1 ADMINISTRATION REGIME ISOFOL MEDICAL AB (SE) 2022-07-06 EP claimed
CN-113336757-B Preparation method of levofolinic acid crystal 南京海纳医药科技股份有限公司 2022-05-13 CN claimed
WO-2022087018-A1 IMPROVED FLUOROURACIL-BASED MULTI-AGENT CHEMOTHERAPY FOR TREATMENT OF METASTATIC COLORECTAL CANCER G1 THERAPEUTICS, INC. (US) 2022-04-28 WO claimed
CN-114324618-A Method for separating and detecting calcium levofolinate intermediate and related substances 重庆华邦制药有限公司 2022-04-12 CN claimed
CN-114280167-A Method for separating and detecting bis (2-hydroxyethyl) disulfide in calcium levofolinate 重庆华邦制药有限公司 2022-04-05 CN claimed
WO-2022066882-A1 METHOD FOR TREATING CANCER WITH A REVERSE TRANSCRIPTASE INHIBITOR ONCOLINEA PHARMACEUTICALS, INC. (US) 2022-03-31 WO claimed
WO-2022058970-A1 KOJIC ACID DERIVATIVE AS SELECTIVE INHIBITOR OF MITOSIS IN COLORECTAL AND GLIOBLASTOMA CANCER CELLS UNIVERSITÀ DEGLI STUDI DI CAGLIARI (IT) 2022-03-24 WO claimed
US-20220024940-A1 STABLE SALT OF 5,10-METHYLENE-(6R)-TETRAHYDROFOLIC ACID Merck & Cie (CH) 2022-01-27 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12564556-B1 Compositions comprising disodium levofolinate FOLR1, FOLR2, SLC19A1 DHFR 7/4885LMNA 2042/4885MTHFD1 8/4885
US-20250127782-A1 METHODS OF TREATING CANCER KRAS, NRAS, EGFR DHFR 9/4885LMNA 3937/4885MTHFD1 29/4885
US-20260124144-A1 COMPOSITIONS COMPRISING DISODIUM LEVOFOLINATE SLC19A1, FOLR1, FOLR2 DHFR 8/4885LMNA 1884/4885MTHFD1 4/4885
US-12539276-B1 Compositions comprising disodium levofolinate SLC19A1, FOLR2, FOLR1 DHFR 8/4885LMNA 2673/4885MTHFD1 7/4885
US-20250215039-A1 NUCLEOSIDES FOR TREATING CANCER UNG, OGG1, NTPCR DHFR 152/4885LMNA 1053/4885MTHFD1 98/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.