SCHEMBL5723792

SCHEMBL5723792

CC(C)(C)[Si](OC1CN(c2nc(C(=O)N3CC(NC(=O)OCc4ccc([N+](=O)[O-])cc4)C3)cs2)C1)(c1ccccc1)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DPP8 Q6V1X1 1/20 0.36
DPP9 Q86TI2 1/20 0.36
TDP1 Q9NUW8 1/20 0.34
PLCG1 P19174 1/20 0.34
ATM Q13315 1/20 0.34
BRD4 O60885 1/20 0.33
BRD2 P25440 1/20 0.33
BRD3 Q15059 1/20 0.33
EPHX1 P07099 2/20 0.33
CCR3 P51677 1/20 0.32
P2RX7 Q99572 1/20 0.32
ROCK2 O75116 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
GAA P10253 1/20 0.32
RAB9A P51151 1/20 0.32
FAAH O00519 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5724334 0.89 CHRM4 (0.39) TDP1PLCG1ATMALDH1A1MAPT
SCHEMBL5724588 0.88 FAAH (0.40) TDP1ATMALDH1A1MAPTFAAH
SCHEMBL5724526 0.87 RAB9A (0.42) TDP1PLCG1ATMCCR3ALDH1A1
SCHEMBL5724203 0.86 DPP8 (0.40) DPP8DPP9TDP1PLCG1ATM
SCHEMBL5724206 0.85 TDP1 (0.34) DPP8DPP9TDP1PLCG1ATM
SCHEMBL7077675 0.85 ENPP2 (0.41)
SCHEMBL5723816 0.85 ENPP2 (0.41)
SCHEMBL5724082 0.85 ENPP2 (0.41)
SCHEMBL5723785 0.85 DPP8 (0.39) DPP8DPP9TDP1PLCG1EPHX1
SCHEMBL5724214 0.84 ENPP2 (0.43) ALDH1A1HPGDFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340757-B1 1-METHYLCARBAPENEM DERIVATIVES SANKYO CO (JP) 2006-10-11 EP disclosed
US-7001897-B2 1-methylcarbapenem derivatives SANKYO COMPANY, LIMITED (JP) 2006-02-21 US disclosed
US-20040014962-A1 1-Methylcarbapenem derivatives SANKYO COMPANY, LIMITED (JP) 2004-01-22 US disclosed
EP-1340757-A1 1-METHYLCARBAPENEM DERIVATIVES Sankyo Company, Limited (JP) 2003-09-03 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040014962-A1 1-Methylcarbapenem derivatives CD14, CPT1A, ACMSD DPP8 1397/4885DPP9 703/4885TDP1 3179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.