SCHEMBL5728055

SCHEMBL5728055

COC(=O)Oc1ccsc1N

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.43
HSD17B10 Q99714 3/20 0.43
HPGD P15428 3/20 0.43
RAB9A P51151 2/20 0.41
NPC1 O15118 1/20 0.41
KMT2A Q03164 7/20 0.41
ALDH1A1 P00352 7/20 0.41
MEN1 O00255 6/20 0.41
MAPT P10636 4/20 0.41
MAPK1 P28482 2/20 0.41
CYP1A2 P05177 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.37
HTT P42858 2/20 0.37
JAK2 O60674 1/20 0.37
GAA P10253 1/20 0.37
LMNA P02545 2/20 0.36
GLA P06280 2/20 0.36
USP2 O75604 1/20 0.36
FLT3 P36888 1/20 0.35
KEAP1 Q14145 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28742962 0.81 ALDH1A1 (0.44) KDM4EHSD17B10HPGDRAB9ANPC1
SCHEMBL11808741 0.79 RAB9A (0.42) KDM4EHSD17B10HPGDRAB9ANPC1
SCHEMBL765304 0.79 KDM4E (0.44) KDM4EHSD17B10HPGDNPC1KMT2A
SCHEMBL18097396 0.79 KMT2A (0.45) HSD17B10HPGDRAB9ANPC1KMT2A
SCHEMBL7079234 0.76 KMT2A (0.40) HSD17B10RAB9ANPC1KMT2AALDH1A1
SCHEMBL4607918 0.74 KDM4E (0.36) KDM4EHSD17B10HPGDRAB9ANPC1
SCHEMBL5728011 0.74 KDM4E (0.44) KDM4EHSD17B10HPGDKMT2AALDH1A1
SCHEMBL5154245 0.73
SCHEMBL5728136 0.73 KDM4E (0.50) KDM4EHSD17B10HPGDKMT2AALDH1A1
SCHEMBL11351584 0.73 KDM4E (0.39) KDM4EHSD17B10HPGDKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1694665-A2 SUBSTITUTED THIOPHENES AiCuris GmbH & Co. KG (DE) 2006-08-30 EP disclosed
WO-2006072348-A2 ALKINYL-SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2006-07-13 WO disclosed
WO-2005063734-A2 SUBSTITUTED THIOPHENES AICURIS GMBH & CO. KG (DE) 2005-07-14 WO disclosed
WO-1997028166-A1 THIENOQUINOLINES BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1997-08-07 WO disclosed