SCHEMBL5740914

SCHEMBL5740914

COC(=O)Oc1cn2ncnc(C3C(=O)Nc4ccc(S(=O)(=O)NCCN5CCOCC5)cc43)c2c1C

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.42
MAPK1 P28482 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
PDE5A O76074 2/20 0.40
MAPK14 Q16539 1/20 0.39
ILK Q13418 1/20 0.38
KDM4E B2RXH2 1/20 0.38
POLB P06746 2/20 0.38
CA12 O43570 1/20 0.37
CA9 Q16790 1/20 0.37
MET P08581 2/20 0.37
NPSR1 Q6W5P4 1/20 0.37
KDR P35968 1/20 0.36
TLR9 Q9NR96 1/20 0.36
TLR8 Q9NR97 1/20 0.36
TLR7 Q9NYK1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740349 0.94 SIGMAR1 (0.40) ALDH1A1MAPK1PDE5AKDRTLR9
SCHEMBL1460905 0.89 MAPK14 (0.44) ALDH1A1MAPK1SMN1; SMN2PDE5AMAPK14
SCHEMBL5739782 0.88 MAPT (0.36) ALDH1A1ILKKDM4EPOLBCA12
SCHEMBL5738334 0.87 KDM4E (0.43) ALDH1A1KDM4E
SCHEMBL5739297 0.84 MAPT (0.34) ALDH1A1MAPK14KDM4EMETKDR
SCHEMBL1461097 0.83 SIGMAR1 (0.39) ALDH1A1MAPK1MAPK14KDR
SCHEMBL5740106 0.82 SYK (0.37) ALDH1A1SMN1; SMN2MAPK14METKDR
SCHEMBL5740762 0.80 KMT2A (0.32) ALDH1A1KDM4EPOLBMETKDR
SCHEMBL7206430 0.78 SMN1; SMN2 (0.46) ALDH1A1MAPK1SMN1; SMN2PDE5AILK
SCHEMBL5739596 0.78 MET (0.39) MAPK14METKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed