SCHEMBL5740349

SCHEMBL5740349

COC(=O)Oc1cn2ncnc(C3C(=O)Nc4ccc(S(=O)(=O)NCCN5CCCC5)cc43)c2c1C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 3/20 0.40
HTR1A P08908 1/20 0.37
ADRA2A P08913 1/20 0.37
PARP1 P09874 3/20 0.36
KDR P35968 2/20 0.35
PDE5A O76074 1/20 0.35
TP53 P04637 1/20 0.35
MAPK1 P28482 1/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
ALDH1A1 P00352 1/20 0.35
MAPT P10636 1/20 0.35
ENPP2 Q13822 1/20 0.35
TLR9 Q9NR96 2/20 0.35
TLR8 Q9NR97 2/20 0.35
TLR7 Q9NYK1 2/20 0.35
PDGFRB P09619 1/20 0.34
SRC P12931 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5740914 0.94 ALDH1A1 (0.42) KDRPDE5AMAPK1ALDH1A1TLR9
SCHEMBL5739782 0.90 MAPT (0.36) KDRTP53ALDH1A1MAPT
SCHEMBL1461097 0.89 SIGMAR1 (0.39) SIGMAR1PARP1KDRTP53MAPK1
SCHEMBL5739297 0.86 MAPT (0.34) KDRTP53ALDH1A1MAPTPDGFRB
SCHEMBL5740106 0.84 SYK (0.37) KDRTP53MEN1KMT2AALDH1A1
SCHEMBL1460905 0.82 MAPK14 (0.44) KDRPDE5AMAPK1ALDH1A1
SCHEMBL5740762 0.82 KMT2A (0.32) KDRTP53MEN1KMT2AALDH1A1
SCHEMBL5738334 0.82 KDM4E (0.43) TP53ALDH1A1MAPT
SCHEMBL5739596 0.79 MET (0.39) KDRPDGFRB
SCHEMBL5740995 0.79 MET (0.33) KDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1183033-B1 PYRROLOTRIAZINE INHIBITORS OF KINASES BRISTOL MYERS SQUIBB CO (US) 2006-03-01 EP claimed