SCHEMBL5742868

SCHEMBL5742868

COC(=O)Cc1cc(Cl)c(Oc2ccccc2)c(Cl)c1

nearest known ligand 0.57

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 17/20 0.57
THRA P10827 15/20 0.57
HSP90AB1 P08238 1/20 0.46
STK39 Q9UEW8 1/20 0.45
RORC P51449 1/20 0.45
LMNA P02545 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7122041 0.86 THRB (0.51) THRBTHRARORC
SCHEMBL3923780 0.86 THRA (0.55) THRBTHRAHSP90AB1LMNA
SCHEMBL5740828 0.82 THRB (0.57) THRBTHRASTK39RORC
SCHEMBL3914044 0.81 THRA (0.50) THRBTHRALMNA
SCHEMBL5388207 0.81 THRB (0.49) THRBTHRAHSP90AB1LMNA
SCHEMBL5385598 0.81 THRB (0.49) THRBTHRAHSP90AB1LMNA
SCHEMBL7114974 0.80 THRB (0.45) THRBTHRARORC
SCHEMBL7122312 0.80 RNF4 (0.47) THRBTHRARORC
SCHEMBL12337187 0.80 THRA (0.48) THRBTHRAHSP90AB1LMNA
SCHEMBL5393176 0.79 THRB (0.57) THRBTHRARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1383729-A4 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORP (US) 2006-04-19 EP disclosed
US-20040267015-A1 Peptide deformylase inhibitors SMITHKLINE BEECHAM CORPORATION 2004-12-30 US disclosed
EP-1383729-A1 PEPTIDE DEFORMYLASE INHIBITORS SmithKline Beecham Corporation (US) 2004-01-28 EP disclosed
WO-2002081426-A1 PEPTIDE DEFORMYLASE INHIBITORS SMITHKLINE BEECHAM CORPORATION (US) 2002-10-17 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040267015-A1 Peptide deformylase inhibitors PDF, PEPD, DPEP1 THRB 2643/4885THRA 3654/4885HSP90AB1 47/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.