SCHEMBL5743009

SCHEMBL5743009

O=C(O)CN(Cc1cccc([N+](=O)[O-])c1)S(=O)(=O)C1(c2c(Cc3ccccc3)oc3ccccc23)C=CC(c2ccccc2)C=C1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.35
PKM P14618 2/20 0.35
KEAP1 Q14145 1/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
LMNA P02545 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
CXCR3 P49682 2/20 0.34
MEN1 O00255 1/20 0.34
POLB P06746 1/20 0.34
KMT2A Q03164 1/20 0.34
MMP1 P03956 1/20 0.33
MMP2 P08253 1/20 0.33
MMP9 P14780 1/20 0.33
MMP8 P22894 1/20 0.33
MMP13 P45452 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5743846 0.88 TAS2R14 (0.36) KEAP1MEN1POLBKMT2APTPN1
SCHEMBL5740580 0.85 PTPN1 (0.36) KEAP1MEN1KMT2APTPN1
SCHEMBL5743012 0.78 PTPN1 (0.35) ALDH1A1PKMKEAP1KDM4EHTT
SCHEMBL4460686 0.75 PTPN1 (0.49) KEAP1PTPN1
SCHEMBL5743318 0.73 KEAP1 (0.37) ALDH1A1KEAP1MEN1POLBKMT2A
SCHEMBL5744955 0.71 MTNR1A (0.35) KEAP1MAPTPTPN1
SCHEMBL4267879 0.68 PTPN1 (0.34) ALDH1A1MMP2MMP13PTPN1
SCHEMBL5742273 0.68 PTPN1 (0.39) PTPN1
SCHEMBL4267916 0.66 ECE1 (0.37) ALDH1A1MEN1KMT2AMMP2MMP13
SCHEMBL5743849 0.65 TAS2R14 (0.35) KEAP1CYP2D6CYP2C9CYP2C19PTPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2006525365-A 2006-11-09 JP claimed
EP-1620422-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B The Institutes for Pharmaceutical Discovery, LLC (US) 2006-02-01 EP claimed
WO-2004099170-A2 PHENYL SUBSTITUTED CARBOXYLIC ACIDS AS INHIBITORS OF PROTEIN TYROSINE PHOSPHATASE-1B THE INSTITUTES FOR PHARMACEUTICAL DISCOVERY, LLC (US) 2004-11-18 WO claimed