SCHEMBL5743796

SCHEMBL5743796

CN(CCO)Cc1ccccc1.Cc1ccc(S(=O)(=O)O)cc1

nearest known ligand 0.50

Known targets — ChEMBL curated mechanism

ABL1BMXBRAFBTKCHRNA4CHRNB2CSNK1EEGFRERBB2F10FLT1FLT3FLT4IGF1RINSRITKJAK3KDRKITOPRM1PARP1PARP2PDGFRBPIK3CDRAF1RETSLC18A2TECTXKdacAdacBdacCftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 9/20 0.50
MCHR1 Q99705 1/20 0.50
SPHK1 Q9NYA1 1/20 0.49
TMEM97 Q5BJF2 1/20 0.47
SIGMAR1 Q99720 1/20 0.47
TAS2R14 Q9NYV8 1/20 0.47
LIMK2 P53671 1/20 0.44
CARM1 Q86X55 1/20 0.44
PRMT6 Q96LA8 1/20 0.44
PRMT8 Q9NR22 1/20 0.44
CNR1 P21554 2/20 0.43
ACKR3 P25106 1/20 0.43
MAPT P10636 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744364 0.92 SIGMAR1 (0.51) CNR2MCHR1TMEM97SIGMAR1TAS2R14
SCHEMBL5530229 0.84 MCHR1 (0.56) CNR2MCHR1TAS2R14LIMK2CNR1
SCHEMBL5745467 0.84 MCHR1 (0.55) CNR2MCHR1TAS2R14CNR1MAPT
SCHEMBL5746050 0.84 CARM1 (0.53) SPHK1TMEM97SIGMAR1CARM1PRMT6
SCHEMBL10719271 0.82 MCHR1 (0.67) CNR2MCHR1TAS2R14CNR1POLB
SCHEMBL135868 0.80 CARM1 (0.64) TMEM97SIGMAR1CARM1PRMT6PRMT8
Phenylethyl Alcohol SCHEMBL28633356 0.79 TDP1 (0.53) CNR2MCHR1MAPTPOLB
SCHEMBL5745728 0.79 MCHR1 (0.52) CNR2MCHR1TAS2R14CNR1
Benzyl Alcohol SCHEMBL1870759 0.79 TSHR (0.52) CNR2MCHR1TAS2R14MAPTPOLB
Dimethylaminoethanol SCHEMBL6669501 0.79 CA2 (0.53) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1288198-B1 PROCESS FOR THE PRODUCTION OF SULFONIC ESTERS KANEKA CORP (JP) 2006-12-20 EP disclosed
US-6992205-B2 Process for the production of sulfonic esters KANEKA CORPORATION (JP) 2006-01-31 US disclosed
US-6864372-B2 Process for the production of sulfonic esters KANEKA CORPORATION (JP) 2005-03-08 US disclosed
US-6794519-B2 Process for the production of sulfonic esters KANEKA CORPORATION (JP) 2004-09-21 US disclosed
US-20030176711-A1 Process for the production of sulfonic esters KANEKA CORPORATION (JP) 2003-09-18 US disclosed
US-20030176713-A1 Reacting an amino alcohol derivative with organic sulfonyl halide in a mixed solvent composed of an aprotic organic solvent and water in presence of a non-water prohibiting inorganic base KANEKA CORPORATION (JP) 2003-09-18 US disclosed
US-20030162966-A1 PROCESS FOR THE PRODUCTION OF SULFONIC ESTERS KANEKA CORPORATION (JP) 2003-08-28 US disclosed
EP-1288198-A1 PROCESS FOR THE PRODUCTION OF SULFONIC ESTERS KANEKA CORPORATION (JP) 2003-03-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030162966-A1 PROCESS FOR THE PRODUCTION OF SULFONIC ESTERS TST, STS, SELENOI CNR2 2713/4885MCHR1 4675/4885SPHK1 2449/4885
US-20030176711-A1 Process for the production of sulfonic esters TST, STS, SELENOI CNR2 2713/4885MCHR1 4675/4885SPHK1 2449/4885
US-20030176713-A1 Reacting an amino alcohol derivative with organic sulfonyl halide in a mixed solvent composed of an aprotic organic solvent and water in presence of a non-water prohibiting inorganic base BRAF, ADH1C, TST CNR2 2565/4885MCHR1 4512/4885SPHK1 2959/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.