SCHEMBL5746141

SCHEMBL5746141

O=C1CC(OCc2cccc3c2Cc2ccccc2-3)C(=O)N1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PNMT P11086 1/20 0.46
TDP2 O95551 2/20 0.36
CASP3 P42574 1/20 0.36
CASP7 P55210 1/20 0.36
CASP9 P55211 1/20 0.36
CASP6 P55212 1/20 0.36
CASP8 Q14790 1/20 0.36
MAP3K14 Q99558 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
CREBBP Q92793 3/20 0.33
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
BRD4 O60885 1/20 0.33
CRBN Q96SW2 3/20 0.32
DDB1 Q16531 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28641177 0.84 PNMT (0.40) PNMTTDP2CASP3CASP7CASP9
SCHEMBL6393796 0.79 PNMT (0.42) PNMTTDP2CASP3CASP7CASP9
SCHEMBL4611913 0.77 NAAA (0.42) PNMTDRD2DRD4DRD3NPC1
SCHEMBL8467847 0.76 PNMT (0.44) PNMTDRD2DRD4DRD3NPC1
SCHEMBL4942730 0.75 GPR39 (0.46) NPC1RAB9ACRBNDDB1IDO1
SCHEMBL1929688 0.71 CRBN (0.44) CREBBPBRD4CRBNDDB1
SCHEMBL10352631 0.71 ALDH1A1 (0.46) TDP2NPC1RAB9ACRBNDDB1
SCHEMBL4816545 0.70 PNMT (0.54) PNMTDRD2DRD4DRD3NPC1
SCHEMBL7538016 0.70 PNMT (0.62) PNMTDRD2DRD4DRD3NPC1
SCHEMBL3979804 0.70 PNMT (0.67) PNMTDRD2DRD4DRD3NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1682540-A1 AZOLIDINECARBONITRILES AND THEIR USE AS DPP-IV INHIBITORS Sankaranarayanan, Alangudi (IN) 2006-07-26 EP disclosed
WO-2005033106-A1 AZOLIDINECARBONITRILES AND THEIR USE AS DPP-IV INHIBITORS SANKARANARAYANAN ALANGUDI (IN) 2005-04-14 WO disclosed