SCHEMBL575227

SCHEMBL575227

O=C(OCCl)Oc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.43
TDP1 Q9NUW8 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ATM Q13315 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
ALOX15 P16050 2/20 0.42
HSD17B10 Q99714 2/20 0.41
HPGD P15428 1/20 0.41
ALDH1A1 P00352 4/20 0.41
CYP19A1 P11511 1/20 0.41
MEN1 O00255 1/20 0.40
HTT P42858 1/20 0.40
GFER P55789 1/20 0.40
KMT2A Q03164 1/20 0.40
RNF4 P78317 1/20 0.40
BCHE P06276 1/20 0.40
USP2 O75604 2/20 0.39
NSD2 O96028 1/20 0.39
MAPK1 P28482 2/20 0.39
TRPA1 O75762 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL575071 0.84 MAPT (0.41) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL27857005 0.83 ELANE (0.37) MAPTATML3MBTL1ALDH1A1USP2
SCHEMBL10025073 0.83 MAPT (0.46) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL8646552 0.83 THRB (0.47) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL22341330 0.82 HSD17B10 (0.49) ALOX15HSD17B10HTTKMT2AUSP2
SCHEMBL6895096 0.81 MAPT (0.44) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL10025075 0.81 MAPT (0.44) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL322125 0.81 MAPT (0.44) MAPTTDP1KDM4EATML3MBTL1
SCHEMBL22228973 0.80 MGLL (0.41) MAPTL3MBTL1MEN1KMT2AMAPK1
SCHEMBL9353461 0.79 TDP1 (0.54) MAPTTDP1KDM4EATML3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 156 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4359419-A1 PRODRUGS WITH 1-(DISULFANYL)ALKYLOXY-CARBONYL UNITS Pharmacytics B.V. (NL) 2024-05-01 EP claimed
CN-117871750-A Method for determining content of lysine 兰州大学 2024-04-12 CN claimed
CN-117858882-A Prodrugs having 1- (disulfanyl) alkoxy-carbonyl units 药物有限公司 2024-04-09 CN claimed
WO-2022271018-A1 PRODRUGS WITH 1-(DISULFANYL)ALKYLOXY-CARBONYL UNITS PHARMACYTICS B.V. (NL) 2022-12-29 WO claimed
US-20260130904-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENE DERIVATIVES AS ANTIPSYCHOTIC AGENTS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2026-05-14 US disclosed
EP-4658663-A2 PRODRUGS OF 4'-SUBSTITUTED NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS Merck Sharp & Dohme LLC (US) 2025-12-10 EP disclosed
US-20240297344-A1 NONAQUEOUS ELECTROLYTE FOR SECONDARY BATTERY AND NONAQUEOUS-ELECTROLYTE SECONDARY BATTERY EMPLOYING THE SAME MITSUBISHI CHEMICAL CORPORATION (JP) 2024-09-05 US disclosed
US-20240287124-A1 PRODRUGS OF 4'-SUBSTITUTED NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2024-08-29 US disclosed
WO-2024163262-A2 PRODRUGS OF 4'-SUBSTITUTED NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2024-08-08 WO disclosed
US-20240217936-A1 5-BENZYLIMIDAZOLE COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF WEST CHINA HOSPITAL, SICHUAN UNIVERSITY (CN) 2024-07-04 US disclosed
EP-4359419-A1 PRODRUGS WITH 1-(DISULFANYL)ALKYLOXY-CARBONYL UNITS Pharmacytics B.V. (NL) 2024-05-01 EP disclosed
CN-117871750-A Method for determining content of lysine 兰州大学 2024-04-12 CN disclosed
EP-1890357-A1 NONAQUEOUS ELECTROLYTE SOLUTION, NONAQUEOUS ELECTROLYTE SECONDARY BATTERY AND CARBONATE COMPOUND Mitsubishi Chemical Corporation (JP) 2008-02-20 EP disclosed
WO-2001056358-A2 ENHANCED PROPERTIED PESTICIDES ROHM AND HAAS COMPANY (US) 2001-08-09 WO disclosed
US-5559266-A Iodinated esters NYCOMED IMAGING AS (NO) 1996-09-24 US disclosed
US-5416223-A Iodinated esters NYCOMED IMAGING AS (NO) 1995-05-16 US disclosed
US-5370861-A Iodinated esters contrast medium and use NYCOMED IMAGING AS (NO) 1994-12-06 US disclosed
EP-0452377-B1 IODINATED ESTERS NYCOMED IMAGING AS (NO) 1994-09-21 EP disclosed
EP-0452377-A1 IODINATED ESTERS. HOLMES MICHAEL JOHN (GB) 1991-10-23 EP disclosed
WO-1990007491-A1 IODINATED ESTERS NYCOMED AS (NO) 1990-07-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240287124-A1 PRODRUGS OF 4'-SUBSTITUTED NUCLEOSIDE REVERSE TRANSCRIPTASE INHIBITORS DNTT, NAPRT, NAMPT MAPT 1204/4885TDP1 254/4885KDM4E 1822/4885
US-20260130904-A1 PIPERAZINE-SUBSTITUTED BENZOTHIOPHENE DERIVATIVES AS ANTIPSYCHOTIC AGENTS EBP, SIGMAR1, EP300 MAPT 703/4885TDP1 3572/4885KDM4E 1490/4885
US-20240217936-A1 5-BENZYLIMIDAZOLE COMPOUND AND PREPARATION METHOD THEREFOR AND USE THEREOF CYP4F11, WASF2, CYP3A5 MAPT 3634/4885TDP1 4531/4885KDM4E 539/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.