SCHEMBL5753860

SCHEMBL5753860

CCOP(=O)(OCC)C(Cc1ccccc1)NS(=O)(=O)c1ccc2nc(SCC3CCCCC3)sc2c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 6/20 0.43
ALDH1A1 P00352 4/20 0.43
HSP90AA1 P07900 1/20 0.43
HPGD P15428 1/20 0.43
TSHR P16473 1/20 0.43
HTT P42858 1/20 0.43
MAPT P10636 6/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GFER P55789 1/20 0.36
PPARA Q07869 1/20 0.36
TP53 P04637 3/20 0.35
POLB P06746 1/20 0.35
THRB P10828 1/20 0.35
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
CYP2C9 P11712 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5756907 0.88 LMNA (0.44) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5756297 0.85 MAPT (0.46) LMNAALDH1A1MAPTSMN1; SMN2GFER
SCHEMBL5754122 0.84 MAPT (0.45) LMNAALDH1A1MAPTSMN1; SMN2GFER
SCHEMBL5755972 0.82 POLB (0.48) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5755993 0.80 MMP2 (0.48) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5757831 0.77 SMN1; SMN2 (0.51) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5757798 0.77 LMNA (0.52) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5755212 0.76 ALDH1A1 (0.51) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5756642 0.74 SMN1; SMN2 (0.50) LMNAALDH1A1HSP90AA1HPGDTSHR
SCHEMBL5756885 0.74 MAPT (0.44) LMNAALDH1A1MAPTSMN1; SMN2GFER

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1208092-B1 SULFONAMIDE DERIVATIVE AS A MATRIX METALLOPROTEINASE INHIBITOR SAMSUNG ELECTRONICS CO LTD (KR) 2006-06-21 EP disclosed
US-6548667-B2 For prevention and treatment of diseases caused by overexpression and overactivation of matrix metalloproteinase SAMSUNG ELECTRONICS CO. LTD. (KR) 2003-04-15 US disclosed
EP-1208092-A4 SULFONAMIDE DERIVATIVE AS A MATRIX METALLOPROTEINASE INHIBITOR SAMSUNG ELECTRONICS CO LTD (KR) 2003-01-02 EP disclosed
US-20020169314-A1 Sulfonamide derivative as a matrix metalloproteinase inhibitor SAMSUNG ELECTRONICS CO. LTD. (KR) 2002-11-14 US disclosed
EP-1208092-A1 SULFONAMIDE DERIVATIVE AS A MATRIX METALLOPROTEINASE INHIBITOR SAMSUNG ELECTRONICS CO., LTD. (KR) 2002-05-29 EP disclosed
WO-2001077092-A1 SULFONAMIDE DERIVATIVE AS A MATRIX METALLOPROTEINASE INHIBITOR SAMSUNG ELECTRONICS CO., LTD. (KR) 2001-10-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020169314-A1 Sulfonamide derivative as a matrix metalloproteinase inhibitor MMP9, MMP3, MMP14 LMNA 1839/4885ALDH1A1 311/4885HSP90AA1 1278/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.