SCHEMBL5756914

SCHEMBL5756914

Fc1cc(C(F)(F)F)ccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 5/20 0.46
TRPV1 Q8NER1 1/20 0.45
IDO1 P14902 2/20 0.44
HSD11B1 P28845 1/20 0.44
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
MCL1 Q07820 3/20 0.41
IL2 P60568 1/20 0.40
MPL P40238 1/20 0.40
MAPT P10636 1/20 0.40
AHR P35869 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30326145 1.00 PDE2A (0.46) PDE2ATRPV1IDO1HSD11B1ALDH1A1
SCHEMBL16971901 0.82 RAPGEF4 (0.37) PDE2ATRPV1HSD11B1ALDH1A1TSHR
SCHEMBL30271700 0.82 RAPGEF4 (0.37) PDE2ATRPV1HSD11B1ALDH1A1TSHR
SCHEMBL29827335 0.81 PDE2A (0.50) PDE2ATRPV1IDO1HSD11B1ALDH1A1
SCHEMBL230800 0.81 PDE2A (0.50) PDE2ATRPV1IDO1HSD11B1ALDH1A1
SCHEMBL8110620 0.80 PDE2A (0.45) PDE2ATRPV1IDO1HSD11B1TSHR
SCHEMBL29402881 0.80 TSHR (0.61) PDE2AALDH1A1TSHRMEN1KMT2A
SCHEMBL980201 0.80 TSHR (0.61) PDE2AALDH1A1TSHRMEN1KMT2A
SCHEMBL3951887 0.79 ESR1 (0.40) HSD11B1TSHRMEN1KMT2A
SCHEMBL530212 0.79 ALDH1A1 (0.41) HSD11B1ALDH1A1TSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 63 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0847977-B1 2,3-DIHALOGENO-6-TRIFLUOROMETHYLBENZENE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME NIPPON SODA CO (JP) 2001-08-29 EP claimed
US-6054605-A CHEMICAL INTERMEDIATE FOR DRUGS, PESTICIDES NIPPON SODA CO., LTD. (JP) 2000-04-25 US claimed
EP-0847977-A1 2,3-DIHALOGENO-6-TRIFLUOROMETHYLBENZENE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME NIPPON SODA CO., LTD. (JP) 1998-06-17 EP claimed
JP-62036336-A None JP disclosed
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON INC (US) 2026-03-12 US disclosed
US-12509474-B2 Inhibitors of complement factors and uses thereof ANNEXON, INC. (US) 2025-12-30 US disclosed
US-12459927-B2 Plasma kallikrein inhibitors MERCK SHARP & DOHME LLC (US) 2025-11-04 US disclosed
US-20240109920-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF ANNEXON, INC. 2024-04-04 US disclosed
US-11814404-B2 Inhibitors of complement factors and uses thereof ANNEXON, INC. (US) 2023-11-14 US disclosed
CN-116947903-A Inhibitors of complement factors and uses thereof 安尼艾克松股份有限公司 2023-10-27 CN disclosed
US-20230286958-A1 PLASMA KALLIKREIN INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-09-14 US disclosed
EP-0159388-A2 Preparation of nuclear chlorinated compounds OCCIDENTAL CHEMICAL CORPORATION (US) 1985-10-30 EP disclosed
EP-0113625-B1 PROCESS FOR THE PREPARATION OF TRIFLUOROMETHYLATED BENZENIC COMPOUNDS RHONE-POULENC CHIMIE (FR) 1985-07-10 EP disclosed
US-4470930-A Preparation of nuclear chlorinated aromatic compounds OCCIDENTAL CHEMICAL CORPORATION (US) 1984-09-11 US disclosed
US-4469893-A Method for the preparation of nitrodiphenyl ethers OCCIDENTAL CHEMICAL CORPORATION (US) 1984-09-04 US disclosed
US-4465508-A Diphenyl ether herbicides IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-08-14 US disclosed
EP-0113625-A1 Process for the preparation of trifluoromethylated benzenic compounds RHONE-POULENC CHIMIE (FR) 1984-07-18 EP disclosed
EP-0023392-B1 DIPHENYL ETHER COMPOUNDS, AND HERBICIDAL COMPOSITIONS AND PROCESSES UTILISING THEM IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1984-06-06 EP disclosed
US-4424396-A ARYL HALIDE, A-AMINOACID OCCIDENTAL CHEMICAL CORPORATION (US) 1984-01-03 US disclosed
EP-0023392-A2 Diphenyl ether compounds, and herbicidal compositions and processes utilising them IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1981-02-04 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240109920-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFB, CFH, C9 PDE2A 1600/4885TRPV1 3867/4885IDO1 1076/4885
US-11814404-B2 Inhibitors of complement factors and uses thereof CFB, CFH, C9 PDE2A 1600/4885TRPV1 3867/4885IDO1 1076/4885
US-12509474-B2 Inhibitors of complement factors and uses thereof SSB, UACA, CFH PDE2A 3080/4885TRPV1 4190/4885IDO1 1123/4885
US-20230286958-A1 PLASMA KALLIKREIN INHIBITORS KLKB1, SERPINE1, KLK5 PDE2A 1472/4885TRPV1 961/4885IDO1 1105/4885
US-20260070932-A1 INHIBITORS OF COMPLEMENT FACTORS AND USES THEREOF CFH, CFB, C5 PDE2A 2194/4885TRPV1 4515/4885IDO1 1216/4885
US-12459927-B2 Plasma kallikrein inhibitors KLKB1, SERPINE1, KLK5 PDE2A 1472/4885TRPV1 961/4885IDO1 1105/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.