SCHEMBL5758191

SCHEMBL5758191

CCS(=O)(=O)c1ccc(CNOC(=O)C(F)(F)F)cc1

nearest known ligand 0.47

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
RORC P51449 19/20 0.47
PSIP1 O75475 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6317990 0.78 HDAC3 (0.54)
SCHEMBL5450071 0.77 CES1 (0.52)
SCHEMBL7734069 0.75 LMNA (0.46)
SCHEMBL20319855 0.72 KMT2A (0.58) RORCPSIP1
SCHEMBL5759432 0.70 RORC (0.59) RORCPSIP1
Trifluoroacetic Acid SCHEMBL5758188 0.70 PSIP1 (0.71) RORCPSIP1
SCHEMBL28253979 0.69 CYP2C9 (0.56) RORCPSIP1
SCHEMBL20943253 0.69 PSIP1 (0.59) RORCPSIP1
SCHEMBL21616664 0.68 RORC (0.53) RORCPSIP1
SCHEMBL19777840 0.68 CA12 (0.66) RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562902-B1 2-PYRIDONE DERIVATIVES AS INHIBITORS OF NEUTROPHILE ELASTASE ASTRAZENECA AB (SE) 2006-05-03 EP disclosed
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase ASRAZENECA AB (SE) 2006-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060035938-A1 2-Pyridone derivatives as inhibitors of neutrophile elastase SERPINB1, ELANE, SERPINE1 RORC 3660/4885PSIP1 3665/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.