SCHEMBL5762863

SCHEMBL5762863

O=C(CCl)NCC(=O)c1cccs1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.66
CASP3 P42574 1/20 0.55
CASP2 P42575 1/20 0.55
ALDH1A1 P00352 4/20 0.55
NPC1 O15118 3/20 0.55
RAB9A P51151 3/20 0.55
POLB P06746 2/20 0.55
MEN1 O00255 1/20 0.55
LMNA P02545 1/20 0.55
KMT2A Q03164 1/20 0.55
KDM4E B2RXH2 1/20 0.51
ERCC5 P28715 1/20 0.51
FEN1 P39748 1/20 0.51
HPGD P15428 4/20 0.49
HDAC1 Q13547 2/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GAA P10253 1/20 0.48
SMN1; SMN2 Q16637 3/20 0.47
MAPT P10636 1/20 0.46
ALOX12 P18054 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30100988 0.81 CASP3 (0.50) GSK3BCASP3CASP2ALDH1A1NPC1
SCHEMBL230036 0.80
SCHEMBL711360 0.76 RAB9A (0.75) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL11084699 0.75 ALDH1A1 (0.62) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL15974627 0.75 ALDH1A1 (0.62) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL11085456 0.75 RAB9A (0.64) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL6771140 0.75 ALDH1A1 (0.67) GSK3BCASP3CASP2ALDH1A1NPC1
Hydrochloric Acid SCHEMBL15974201 0.74 ALDH1A1 (0.60) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL960143 0.73 ALDH1A1 (0.77) GSK3BALDH1A1NPC1RAB9APOLB
SCHEMBL8505274 0.72 ALDH1A1 (0.58) GSK3BALDH1A1NPC1RAB9APOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1270571-B1 Heterocyclic compounds, their production and use TAKEDA PHARMACEUTICAL (JP) 2006-09-06 EP disclosed
EP-1270571-A1 Heterocyclic compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2003-01-02 EP disclosed
US-6211215-B1 AROMATIC HETEROCYCLIC COMPOUND WITH AZOLE COMPOUND TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-04-03 US disclosed
EP-0912562-A1 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1999-05-06 EP disclosed
WO-1998003505-A2 HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-01-29 WO disclosed