SCHEMBL5763645

SCHEMBL5763645

O=C(c1ccc(CNc2c(Cl)ccc3c2CCC(C(=O)C(F)(F)F)CN3)cc1)C1CCCCC1

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.33
KCNH2 Q12809 1/20 0.32
HDAC6 Q9UBN7 2/20 0.32
SSTR3 P32745 2/20 0.32
SRD5A2 P31213 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
POLB P06746 1/20 0.31
MAPT P10636 1/20 0.31
RORC P51449 1/20 0.31
SMN1; SMN2 Q16637 2/20 0.30
HPGD P15428 1/20 0.30
LMNA P02545 1/20 0.30
HTT P42858 1/20 0.30
P2RX7 Q99572 1/20 0.30
MLYCD O95822 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5767548 0.89 RAB9A (0.33) ALDH1A1POLBSMN1; SMN2
SCHEMBL5736358 0.87 ALDH1A1 (0.37) ALDH1A1MAPTLMNAHTT
SCHEMBL5755390 0.86 P2RX7 (0.32) RORCP2RX7
SCHEMBL5756968 0.83 CRHR1 (0.39) ALDH1A1SMN1; SMN2HPGD
SCHEMBL4765020 0.80 POLB (0.33) POLBMAPTHPGDP2RX7
Succinic Acid SCHEMBL5757273 0.79 HRH3 (0.36) ALDH1A1KCNH2HDAC6SSTR3SRD5A2
SCHEMBL5733066 0.79 P2RX7 (0.33) P2RX7
SCHEMBL5754230 0.77 WDR5 (0.33) P2RX7
SCHEMBL5756080 0.77 KCNH2 (0.40) KCNH2
SCHEMBL4775977 0.76 TBK1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1720836-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO [D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2006-11-15 EP disclosed
WO-2005082859-A1 6-SUBSTITUTED 2,3,4,5-TETRAHYDRO-1H-BENZO[D]AZEPINES AS 5-HT2C RECEPTOR AGONISTS ELI LILLY AND COMPANY (US) 2005-09-09 WO disclosed