SCHEMBL5766444

SCHEMBL5766444

COc1ccc2c(c1)SCc1cccc(N)c1C2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.46
HTT P42858 1/20 0.46
MAPK14 Q16539 4/20 0.45
CA12 O43570 6/20 0.43
CA9 Q16790 6/20 0.43
CA1 P00915 5/20 0.43
CA2 P00918 5/20 0.43
CA3 P07451 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA13 Q8N1Q1 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
EGFR P00533 1/20 0.43
HSD17B3 P37058 1/20 0.43
MAOA P21397 1/20 0.43
MAOB P27338 1/20 0.43
LMNA P02545 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5763637 0.81 ACHE (0.52) KDM4EHTTCA12CA9CA1
SCHEMBL29853726 0.75 CA12 (0.53) KDM4EHTTCA12CA9CA1
SCHEMBL26768607 0.75 CA12 (0.53) KDM4EHTTCA12CA9CA1
SCHEMBL19334753 0.73 ALDH1A1 (0.39) KDM4EHTTMAPK14EGFRHSD17B3
SCHEMBL5765246 0.73 PDK1 (0.48) CA12CA9CA1CA2HSD17B3
SCHEMBL68574 0.72 KDM4E (0.71) KDM4EHTTCA12CA9CA1
SCHEMBL15143531 0.69 MAPT (0.50) KDM4EHTTCA9CA1CA2
SCHEMBL11481280 0.69 MAPT (0.57) KDM4EHTTMAPK14HSD17B3MAOA
SCHEMBL86336 0.69 MAPT (0.50) KDM4EMAPK14CA12CA9CA1
SCHEMBL22259137 0.68 CYP26A1 (0.59) KDM4EHTTMAPK14LMNAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979821-B1 TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO KK (JP) 2006-09-13 EP disclosed
US-6211227-B1 SULFUR CONTAINING TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO CO., LTD. (JP) 2001-04-03 US disclosed
EP-0979821-A1 TRICYCLIC COMPOUNDS KYOWA HAKKO KOGYO CO., LTD. (JP) 2000-02-16 EP disclosed