SCHEMBL5767698

SCHEMBL5767698

CCC(CC)(C(=O)O)c1cc(C(F)(F)F)cc(C(F)(F)F)c1

nearest known ligand 0.47

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.47
ALDH1A1 P00352 2/20 0.45
RXRA P19793 4/20 0.42
RXRB P28702 4/20 0.42
RXRG P48443 3/20 0.42
LMNA P02545 1/20 0.42
TACR1 P25103 3/20 0.42
MAPT P10636 1/20 0.42
AKR1C3 P42330 1/20 0.39
AKR1C2 P52895 1/20 0.39
GPR35 Q9HC97 1/20 0.39
P2RX1 P51575 1/20 0.39
NOTUM Q6P988 1/20 0.39
AGBL2 Q5U5Z8 1/20 0.38
ACP1 P24666 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3355856 0.84 CES2 (0.47) CES2ALDH1A1LMNA
SCHEMBL5764207 0.79 NOTUM (0.46) CES2ALDH1A1LMNAMAPTGPR35
SCHEMBL14372751 0.78 GPR35 (0.46) CES2ALDH1A1LMNAMAPTGPR35
Hydrochloric Acid SCHEMBL4499764 0.76 ALDH1A1 (0.43) CES2ALDH1A1MAPTNOTUM
SCHEMBL25460762 0.73 NOTUM (0.37) RXRARXRBRXRGNOTUMACP1
SCHEMBL10898859 0.73 MEN1 (0.42) CES2LMNA
SCHEMBL504013 0.72 ALDH1A1 (0.57) ALDH1A1LMNAMAPT
SCHEMBL531511 0.72 CES2 (0.52) CES2ALDH1A1RXRARXRBRXRG
SCHEMBL4028192 0.72 APP (0.53) CES2ALDH1A1RXRARXRBRXRG
SCHEMBL30221940 0.72 CES2 (0.47) CES2ALDH1A1RXRARXRBRXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286967-B1 CYCLOHEXANE DERIVATIVES AND THEIR USE AS THERAPEUTIC AGENTS MERCK SHARP & DOHME (GB) 2006-09-27 EP disclosed
US-7105507-B2 Cyclohexane derivatives and their use as therapeutic agents MERCK SHARP & DOHME LIMITED (GB) 2006-09-12 US disclosed
US-20030236250-A1 Cyclohexane derivatives and their use as therapeutic agents MERCK SHARP & DOHME LTD. (GB) 2003-12-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030236250-A1 Cyclohexane derivatives and their use as therapeutic agents CNR2, CNR1, HTR1A CES2 811/4885ALDH1A1 1452/4885RXRA 908/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.