SCHEMBL5772801

SCHEMBL5772801

Cc1nc(C2=CNCC2)c2nc(-c3ccc(Cl)c(Cl)c3)cc-2[nH]1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 3/20 0.36
NPY5R Q15761 5/20 0.33
NPC1 O15118 2/20 0.33
NFKB1 P19838 2/20 0.33
RAB9A P51151 2/20 0.33
NFKB2 Q00653 2/20 0.33
RELA Q04206 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MAPT P10636 2/20 0.32
ALDH1A1 P00352 2/20 0.32
NPFFR1 Q9GZQ6 1/20 0.32
NPFFR2 Q9Y5X5 1/20 0.32
HPGD P15428 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
KMT2A Q03164 2/20 0.31
PIM1 P11309 1/20 0.31
NOTUM Q6P988 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5778148 0.98 KMO (0.34) KMONPY5RNPC1NFKB1RAB9A
SCHEMBL5772019 0.85 TGFBR1 (0.39) NPY5R
SCHEMBL5773678 0.83 RAD51 (0.36) NPC1RAB9AMAPTKMT2AMEN1
Hydrochloric Acid SCHEMBL5777028 0.83 HTR2C (0.38) NPY5R
Hydrochloric Acid SCHEMBL5773419 0.81 RAD51 (0.34) NPC1RAB9AMAPTKMT2AMEN1
SCHEMBL5772572 0.79 KMO (0.43) KMONPY5RNPC1RAB9AMAPT
SCHEMBL5772104 0.78 XDH (0.41) NPY5RKDM4EALDH1A1HPGDKMT2A
SCHEMBL5775574 0.76 KMO (0.44) KMONPY5RNPC1RAB9AKDM4E
Hydrochloric Acid SCHEMBL5774377 0.76 HTR2C (0.41) NPY5RKDM4EALDH1A1HPGDKMT2A
SCHEMBL5772805 0.73 HRH4 (0.39) KMONPY5RNPC1NFKB1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed