SCHEMBL5773678

SCHEMBL5773678

Cc1nc(C2=CNCC2)c2nc(-c3ccc(F)cc3)cc-2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAD51 Q06609 1/20 0.36
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
ALOX15 P16050 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
MAPK14 Q16539 2/20 0.33
GSK3B P49841 1/20 0.33
THRB P10828 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
SCN9A Q15858 1/20 0.32
MAPKAPK2 P49137 1/20 0.32
MAPT P10636 3/20 0.31
GCGR P47871 1/20 0.31
ADORA2A P29274 1/20 0.31
ADORA1 P30542 1/20 0.31
MGAM O43451 1/20 0.31
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5773419 0.98 RAD51 (0.34) RAD51MEN1NPC1ALOX15RAB9A
SCHEMBL5772801 0.83 KMO (0.36) MEN1NPC1RAB9AKMT2AMAPT
Hydrochloric Acid SCHEMBL5778148 0.81 KMO (0.34) NPC1RAB9AKMT2AMAPT
SCHEMBL5772019 0.80 TGFBR1 (0.39) HTR2CMAPKAPK2MGAMGAASI
SCHEMBL5772104 0.80 XDH (0.41) MEN1KMT2AHTR2C
Hydrochloric Acid SCHEMBL5777028 0.78 HTR2C (0.38) HTR2CMAPKAPK2MGAMGAASI
Hydrochloric Acid SCHEMBL5774377 0.78 HTR2C (0.41) MEN1KMT2AHTR2C
SCHEMBL5774514 0.75 MEN1 (0.44) RAD51MEN1NPC1ALOX15RAB9A
SCHEMBL5772074 0.75 RAD51 (0.41) RAD51MEN1NPC1ALOX15RAB9A
SCHEMBL5773685 0.72 NPY5R (0.40) RAD51THRBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1054887-B1 BICYCLIC PYRIDINE AND PYRIMIDINE DERIVATIVES AS NEUROPEPTIDE Y RECEPTOR ANTAGONISTS AMGEN INC (US) 2006-04-12 EP claimed
US-6187777-B1 PYRROLO(3,2-D)PYRIMIDINE DERIVATIVES; NEUROPEPTIDE Y AND CORTICOTROPIN RELEASING FACTOR MODULATORS; DIETETICS; ANTIDIABETIC, ANTIINFLAMMATORY, AND ANTITUMOR AGENTS AMGEN INC. 2001-02-13 US claimed