SCHEMBL5774728

SCHEMBL5774728

CC1(c2ccccc2)CC(Nc2c(Cl)cc(Cl)cc2Cl)C(=O)O1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 5/20 0.40
HSD11B1 P28845 8/20 0.39
LDHA P00338 1/20 0.36
DRD1 P21728 2/20 0.34
TNKS O95271 1/20 0.32
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HTR1A P08908 1/20 0.31
HTR2A P28223 1/20 0.31
HTR7 P34969 1/20 0.31
HCAR3 P49019 1/20 0.31
HCAR2 Q8TDS4 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5777138 0.86 HSD11B1 (0.39) HTR6HSD11B1LDHATNKSLMNA
SCHEMBL5775190 0.80 GSK3B (0.35) HSD11B1
SCHEMBL5776425 0.80 HSD11B1 (0.39) HSD11B1LMNATP53HTTNPSR1
SCHEMBL5778899 0.80 THRB (0.38) HSD11B1LDHATP53ALDH1A1KDM4E
SCHEMBL5776022 0.79 NPSR1 (0.41) HSD11B1LMNATP53HTTNPSR1
SCHEMBL5773915 0.79 HSD11B1 (0.43) HSD11B1ALDH1A1KDM4EHCAR3HCAR2
SCHEMBL5778953 0.78 ALDH1A1 (0.41) HSD11B1LDHAALDH1A1KDM4EGAA
SCHEMBL5777244 0.78 P2RX7 (0.36) HTR6HSD11B1
SCHEMBL5775030 0.77 HTR6 (0.34) HTR6HSD11B1ALDH1A1
SCHEMBL5775758 0.77 HSD11B1 (0.38) HSD11B1HCAR3HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1406888-B1 SUBSTITUTED Y-LACTONE COMPOUNDS SERVING AS NMDA ANTAGONISTS GRUENENTHAL GMBH (DE) 2006-05-24 EP disclosed