SCHEMBL5776448

SCHEMBL5776448

COc1ccc2nccc(NC(=O)ON3CCN(CC(=O)c4ccc5c(c4)NC(=O)CO5)CC3)c2n1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.46
HTR1A P08908 1/20 0.46
HTR1B P28222 1/20 0.46
KCNH2 Q12809 6/20 0.42
ALDH1A1 P00352 4/20 0.41
MAPT P10636 7/20 0.40
POLB P06746 2/20 0.40
RXFP1 Q9HBX9 2/20 0.40
USP2 O75604 1/20 0.40
BLM P54132 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7099789 0.90 HTR1D (0.47) HTR1DHTR1AHTR1BKCNH2ALDH1A1
SCHEMBL5764977 0.89 HTR1D (0.53) HTR1DHTR1AHTR1BKCNH2ALDH1A1
SCHEMBL5771874 0.86 KCNH2 (0.41) KCNH2
SCHEMBL5750593 0.79 HTR1D (0.46) HTR1DHTR1AHTR1BKCNH2ALDH1A1
SCHEMBL5764950 0.76 HTR1A (0.51) HTR1DHTR1AHTR1BKCNH2
SCHEMBL5765233 0.75 SLC2A1 (0.43) HTR1DHTR1AKCNH2
SCHEMBL5765739 0.75 ALDH1A1 (0.40) HTR1DHTR1AHTR1BKCNH2ALDH1A1
SCHEMBL5751074 0.75 NPC1 (0.41) KCNH2ALDH1A1POLB
SCHEMBL14573146 0.75 KCNH2 (0.49) HTR1DHTR1AHTR1BKCNH2
SCHEMBL5762645 0.74 KCNH2 (0.53) KCNH2ALDH1A1POLBKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1343780-B1 PIPERAZINE DERIVATIVES FOR TREATMENT OF BACTERIAL INFECTIONS SMITHKLINE BEECHAM PLC (GB) 2006-09-20 EP claimed