SCHEMBL5793789

SCHEMBL5793789

COc1cccc2cc(C(=O)NN(CC(C)(C)C)c3ccnc(C#N)n3)oc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.43
RECQL P46063 1/20 0.43
CTSK P43235 3/20 0.43
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
BMP1 P13497 4/20 0.41
RXFP1 Q9HBX9 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KDM4E B2RXH2 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
MEN1 O00255 1/20 0.40
HPGD P15428 1/20 0.40
MAPT P10636 3/20 0.40
CTSL P07711 1/20 0.40
CTSB P07858 1/20 0.40
CTSS P25774 1/20 0.40
CTSC P53634 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8270695 0.88 LMNA (0.43) LMNARECQLALDH1A1KMT2AHDAC1
SCHEMBL8269391 0.88 LMNA (0.46) LMNARECQLALDH1A1KMT2AHDAC1
Trifluoroacetic Acid SCHEMBL5791293 0.85 BMP1 (0.41) LMNARECQLALDH1A1KMT2AHDAC1
SCHEMBL5794707 0.81 LMNA (0.43) LMNARECQLCTSKALDH1A1KMT2A
SCHEMBL5791966 0.79 CTSK (0.45) CTSKALDH1A1KMT2ANPC1RAB9A
SCHEMBL8268844 0.76 CTSK (0.45) LMNARECQLCTSKALDH1A1KMT2A
SCHEMBL8270702 0.76 NPC1 (0.46) LMNACTSKALDH1A1KMT2ANPC1
SCHEMBL8271448 0.75 CTSK (0.46) CTSKKMT2AHDAC1NPC1RAB9A
SCHEMBL8245768 0.74 CTSL (0.53) LMNARECQLCTSKALDH1A1KMT2A
SCHEMBL5791503 0.74 CTSK (0.47) CTSKALDH1A1HDAC1HDAC2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006027211-A1 2,4-SUBSTITUTED PYRIMIDINES AS CYSTEINE PROTEASE INHIBITORS GLAXO GROUP LIMITED (GB) 2006-03-16 WO disclosed