SCHEMBL5801209

SCHEMBL5801209

NC(=O)C(c1ccccc1)N(C(N)=O)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TRPM8 Q7Z2W7 14/20 0.47
MDM2 Q00987 1/20 0.45
CES2 O00748 1/20 0.41
CES1 P23141 1/20 0.41
NR1I2 O75469 2/20 0.39
KDM4E B2RXH2 1/20 0.39
GAA P10253 1/20 0.39
ALOX5 P09917 1/20 0.39
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
ALOX15 P16050 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EPHX1 P07099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3568466 0.91 TRPM8 (0.41) TRPM8MDM2CES2CES1KDM4E
SCHEMBL5802781 0.88 TRPM8 (0.45) TRPM8MDM2CES2CES1NR1I2
SCHEMBL5819200 0.83 ALDH1A1 (0.56) TRPM8MDM2GAANPC1ALDH1A1
SCHEMBL5801133 0.82 MDM2 (0.39) MDM2CES2CES1NR1I2KDM4E
SCHEMBL5819192 0.80 NPC1 (0.49) TRPM8MDM2GAANPC1ALDH1A1
SCHEMBL5803975 0.80 MDM2 (0.34) TRPM8MDM2CES2CES1NPC1
SCHEMBL7560686 0.78 ALOX5 (0.44) TRPM8NR1I2ALOX5ALDH1A1MAPT
SCHEMBL3563022 0.78 MDM2 (0.41) MDM2CES2CES1NR1I2KDM4E
SCHEMBL3563412 0.76 PPARA (0.38) MDM2CES2CES1GAANPC1
SCHEMBL3569300 0.76 CNR2 (0.41) MDM2CES2CES1GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006063113-A2 UREAS AS FACTOR XA INHIBITORS PORTOLA PHARMACEUTICALS, INC. (US) 2006-06-15 WO claimed