SCHEMBL5801633

SCHEMBL5801633

C=C(C[C@H](N[S+]([O-])C(C)(C)C)C(=O)OCC)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.41
PPARG P37231 1/20 0.41
PTPN1 P18031 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
POLB P06746 2/20 0.35
MAPT P10636 4/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
HSP90AA1 P07900 1/20 0.34
CRHBP P24387 1/20 0.34
KMT2A Q03164 1/20 0.34
CRHR2 Q13324 1/20 0.34
GAA P10253 2/20 0.34
TRPV1 Q8NER1 1/20 0.34
ALDH1A1 P00352 2/20 0.33
CYP1A1 P04798 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5797762 1.00 EPHX2 (0.41) EPHX2PPARGPTPN1NPSR1NPC1
SCHEMBL5797287 0.89 GPR35 (0.35) EPHX2PPARGNPSR1SMN1; SMN2POLB
SCHEMBL5797971 0.89 GPR35 (0.35) EPHX2PPARGNPSR1SMN1; SMN2POLB
SCHEMBL5797834 0.89 KMT2A (0.37) NPC1RAB9APOLBMAPTMEN1
SCHEMBL5820016 0.89 KMT2A (0.37) NPC1RAB9APOLBMAPTMEN1
SCHEMBL5799304 0.86 KMT2A (0.43) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL5798028 0.86 KMT2A (0.43) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL5801142 0.86 CYP26A1 (0.40) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL5800376 0.86 CYP26A1 (0.40) NPC1RAB9ASMN1; SMN2MAPTMEN1
SCHEMBL5814731 0.83 ALDH1A1 (0.40) NPC1RAB9ASMN1; SMN2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006030208-A1 AMINO ACID UNIVERSITY OF LEEDS (GB) 2006-03-23 WO claimed
WO-2006030208-A1 AMINO ACID UNIVERSITY OF LEEDS (GB) 2006-03-23 WO disclosed