SCHEMBL581713

SCHEMBL581713

COc1ccc(Cc2c(F)ccc(C(N)=O)c2NC2CCOCC2)cc1OC

nearest known ligand 0.43

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSD P07339 5/20 0.43
JAK1 P23458 5/20 0.41
JAK3 P52333 5/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
HTT P42858 1/20 0.40
KCNH2 Q12809 2/20 0.40
ALDH1A1 P00352 2/20 0.39
ATM Q13315 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
ROCK2 O75116 1/20 0.38
ROCK1 Q13464 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL583113 0.82 CTSD (0.46) CTSDJAK1JAK3MEN1KMT2A
SCHEMBL4582130 0.75 TUBB4A (0.42) CTSDJAK1JAK3MEN1KMT2A
SCHEMBL17766573 0.74 JAK1 (0.47) JAK1JAK3KCNH2ATMROCK2
SCHEMBL581712 0.71 HDAC3 (0.52) KMT2AALDH1A1MAPK1
SCHEMBL6153322 0.71 FLT3 (0.47) JAK1JAK3MEN1KMT2A
SCHEMBL581422 0.71 MEN1 (0.40) JAK1JAK3MEN1KMT2AALDH1A1
SCHEMBL17766551 0.69 JAK1 (0.53) JAK1JAK3KCNH2ATMROCK2
SCHEMBL3683008 0.69 PDE4B (0.47) JAK1JAK3KCNH2ATM
SCHEMBL17766577 0.68 MAP2K2 (0.42) JAK1JAK3KCNH2ATMROCK2
SCHEMBL2684142 0.68 NPC1 (0.55) CTSDHTTALDH1A1L3MBTL1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417130-A2 QUINAZOLINEDIONE DERIVATIVES, PREPARATION THEREOF AND VARIOUS THERAPEUTIC USES THEREOF SANOFI (FR) 2012-02-15 EP disclosed