SCHEMBL583113

SCHEMBL583113

COc1ccc(Cc2cccc(C(N)=O)c2NC2CCOCC2)cc1OC

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CTSD P07339 4/20 0.46
HTT P42858 1/20 0.41
ALDH1A1 P00352 2/20 0.40
JAK1 P23458 4/20 0.40
JAK3 P52333 4/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
HTR2B P41595 1/20 0.40
GAA P10253 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
RAB9A P51151 1/20 0.39
PDE4B Q07343 1/20 0.39
APEX1 P27695 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL581422 0.88 MEN1 (0.40) ALDH1A1JAK1JAK3HTR2AHTR2C
SCHEMBL581713 0.82 CTSD (0.43) CTSDHTTALDH1A1JAK1JAK3
SCHEMBL582321 0.75 CA2 (0.54) HTTALDH1A1GAAMEN1KMT2A
SCHEMBL4582130 0.75 TUBB4A (0.42) CTSDHTTALDH1A1JAK1JAK3
SCHEMBL29229026 0.73 CXCR2 (0.51) ALDH1A1JAK1JAK3PDE4B
SCHEMBL583112 0.73 APEX1 (0.53) ALDH1A1GAAMEN1KMT2ARAB9A
SCHEMBL17766551 0.71 JAK1 (0.53) JAK1JAK3PDE4B
SCHEMBL28811459 0.71 CA2 (0.45) HTTALDH1A1GAAMEN1KMT2A
SCHEMBL6153322 0.70 FLT3 (0.47) JAK1JAK3GAAMEN1KMT2A
SCHEMBL4580646 0.69 CTSD (0.42) CTSDALDH1A1JAK1JAK3MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2417130-A2 QUINAZOLINEDIONE DERIVATIVES, PREPARATION THEREOF AND VARIOUS THERAPEUTIC USES THEREOF SANOFI (FR) 2012-02-15 EP disclosed