SCHEMBL5820519

SCHEMBL5820519

CC(C)Oc1ccccc1C1CCN(Cc2cccc(C(=O)N3CCc4ccc(NCc5ccccc5F)cc43)c2)CC1

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 3/20 0.54
ADRA1D P25100 2/20 0.54
ADRA1A P35348 2/20 0.54
ADRA1B P35368 2/20 0.54
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
DRD2 P14416 1/20 0.42
HTR1B P28222 1/20 0.42
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5820685 0.88 ADRA1D (0.55) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5814914 0.84 HTR1A (0.75) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5899207 0.83 HTR1A (0.62) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5820590 0.81 MEN1 (0.55) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5899201 0.75 MEN1 (0.63) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5805494 0.74 MEN1 (0.51) MEN1KMT2ADRD2
SCHEMBL9540927 0.73 HTR1A (0.70) HTR1AADRA1DADRA1AADRA1BMEN1
Hydrochloric Acid SCHEMBL7648536 0.73 HTR1A (0.69) HTR1AADRA1DADRA1AADRA1BMEN1
SCHEMBL5819994 0.72 HTR1A (0.72) HTR1AADRA1DADRA1AADRA1BDRD2
SCHEMBL5813989 0.72 ALDH1A1 (0.50) MEN1KMT2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006088954-A1 DIHYDROINDOLYL METHANONES AS ALPHA 1A/1D ADRENORECEPTOR MODULATORS FOR THE TREATMENT OF BENIGN PROSTATIC HYPERTROPHY AND LOWER URINARY TRACT SYMPTOMS JANSSEN PHARMACEUTICA, N.V. (BE) 2006-08-24 WO disclosed